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Patent # Description
2016/0122359 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF
Disclosed are compounds having enhanced potency in the modulation of NMD A receptor activity. Such compounds are contemplated for use in the treatment of...
2016/0122358 NOVEL SUBSTITUTED PYRAZOLO-PIPERAZINES AS CASEIN KINASE 1 D/E INHIBITORS
The invention provides compounds of Formula (I): ##STR00001## and pharmaceutically acceptable salts thereof. The compounds of Formula (I) inhibit protein kinase...
2016/0122357 PYRIMIDO-DIAZEPINONE KINASE SCAFFOLD COMPOUNDS AND METHODS OF TREATING DISORDERS
The present invention relates to novel pyrimido-diazepinone compounds, methods of modulating protein kinases, including MPS1 (TTK), ERK5 (BMK1, MAPK7), polo...
2016/0122356 METHODS FOR THE PREPARATION OF RIBOSIDES
Provided are methods of preparing compounds and pharmaceutical compositions for treating Filoviridae virus infections The compounds, compositions, and methods...
2016/0122355 CRYSTALLINE FORMS OF PEMETREXED DIACID AND MANUFACTURING PROCESSES THEREFOR
Crystalline forms of pemetrexed diacid are provided (Forms 1 and 2) which are readily produced for either laboratory-scale or industrial scale. Processes for...
2016/0122354 PROCESS FOR THE PREPARATION OF (3R,4R)-4-METHYL-3-(METHYL-7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL-AMINO)- ...
The present invention relates to an improved 7H-pyrrolo[2,3-d]pyrimidin-4-yl-amino)-.beta.-oxo-1-piperidine propanenitrile compound of formula-1 and its...
2016/0122353 HETEROCYCLIC COMPOUNDS AS PEST CONTROL AGENTS
The present application relates to the use of known and novel heterocyclic compounds for controlling animal pests, to novel heterocyclic compounds, to...
2016/0122352 POLYMORPHS
The invention relates to polymorphous crystal modifications of a DPP-IV inhibitor, the preparation thereof and the use thereof for preparing a medicament.
2016/0122351 Substituted Pyrimidinium Compounds and Derivatives for Combating Animal Pests
Substituted pyrimidinium compounds of the general formula (I) and their uses for combating animal pests The present invention relates to substituted pyrimidinium...
2016/0122350 PROCESS FOR THE PREPARATION OF CHIRAL TERT-BUTYL ...
A process for the preparation of N-protected 6-(piperidin-4-ylcarbamoyl)piperidin-3-yl sulfonates of Formula (III): which comprises contacting a lactone of...
2016/0122349 MORPHINAN DERIVATIVE
The present invention relates to a morphinan derivative represented by the following general formula (I), wherein R.sup.1 represents hydrogen, C.sub.1-6 alkyl,...
2016/0122348 COMPOUNDS AND ANTI-TUMOR NQO1 SUBSTRATES
Compounds of Formula (I) can be selectively lethal toward a variety of different cancer cell types. The compounds are useful for the management, treatment,...
2016/0122347 4,6-DIAMINOPYRIMIDINE STIMULATORS OF SOLUBLE GUANYLATE CYCLASE
The present invention relates to new 4,6-diaminopyrimidine stimulators of soluble guanylate cyclase, pharmaceutical compositions thereof, and methods of use...
2016/0122346 NOVEL 1,3-DIHYDRO-2H-BENZIMIDAZOL-2-ONE DERIVATIVES SUBSTITUTED WITH HETEROCYCLES AS RESPIRATORY SYNCYTIAL...
The present invention is concerned with novel 1,3-dihydro-2H-benzimidazol-2-one derivatives substituted with heterocycles having formula (I) ##STR00001## ...
2016/0122345 DIHYDROPYRROLOPYRIDINE INHIBITORS OF ROR-GAMMA
Provided are novel compounds of Formula (I): ##STR00001## pharmaceutically acceptable salts thereof, and pharmaceutical compositions thereof, which are useful in...
2016/0122344 Novel 6,7-dihydrobenzo[a]quinolizin-2-one derivatives for the treatment and prophylaxis of hepatitis B virus...
The invention provides novel compounds having the general formula: ##STR00001## wherein R.sup.1 to R.sup.6, W and X are as described herein and their ...
2016/0122343 Novel Pyridopyrimidinone Compounds for Modulating the Catalytic Activity of Histone Lysine Demethylases (KDMs)
The present invention provides a compound of Formula (I) being capable of modulating the activity of histone lysine demethylase (KDM), pharmaceutical...
2016/0122342 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS
This invention relates to novel compounds according to Formula (I) which are inhibitors of Enhancer of Zeste Homolog 2 (EZH2), to pharmaceutical compositions...
2016/0122341 3-ARYL-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINES AND THEIR USE
The present application relates to novel 3-aryl-substituted imidazo[1,2-a]pyridines, to processes for preparation thereof, to the use thereof, alone or in...
2016/0122340 HISTONE DEACETYLASE INHIBITORS BASED ON DERIVATIVES OF TRICYCLIC POLYHYDROACRIDINE AND ANALOGS POSSESSING FUSED...
The present invention refers to compounds of formula (I): ##STR00001## as well as to a method for their preparation, pharmaceutical compositions comprising the...
2016/0122339 [1,2,4] TRIAZOL [4,3-A] PYRIDINE DERIVATIVE, PREPARATION METHOD THEREFOR OR MEDICAL APPLICATION THEREOF
Provided are [1,2,4]triazol[4,3-a]pyridine derivatives as shown in the general formula (I), a preparation method therefor, and a pharmaceutical composition...
2016/0122338 NOVEL PHOTOCHROMIC TETRAHYDROINDOLIZINES
Photochromic tetrahydroindolizines (THIs) bearing dihydroisoquinoline derivatives as heterocyclic bases and central fluorene groups have been synthesized via...
2016/0122337 2-HETEROARYL CARBOXAMIDES
The invention relates to novel 2-heteroaryl carboxamides and to the use thereof for producing medicaments for the treatment and/or prophylaxis of diseases and...
2016/0122336 TRIFLUOROMETHYL ALCOHOLS AS MODULATORS OF RORyt
The present invention comprises compounds of Formula I. ##STR00001## wherein: X, A.sup.1, A.sup.2, A.sup.3, A.sup.4, R.sup.1, R.sup.2, and R.sup.3 are defined in...
2016/0122335 AMIDE SUBSTITUTED THIAZOLES AS MODULATORS OF RORyt
The present invention comprises compounds of Formula I. ##STR00001## wherein: R.sup.1, R.sup.2, R.sup.3, R.sup.5, A.sup.1, A.sup.2, and ##STR00002## are defined in...
2016/0122334 INHIBITORS OF C-FMS KINASE
The invention is directed to compounds of Formula I: ##STR00001## wherein Z, X, J, R.sup.2 and W are set forth in the specification, as well as solvates,...
2016/0122333 MULTISUBSTITUTED AROMATIC COMPOUNDS AS INHIBITORS OF THROMBIN
There are provided inter alia multisubstituted aromatic compounds useful for the inhibition of thrombin, which compounds include substituted pyrazolyl or...
2016/0122332 COMPOSITIONS AND METHODS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS
The invention relates to the compounds of formula I and formula IA or its pharmaceutical acceptable salts, as well as polymorphs, solvates, enantiomers,...
2016/0122331 SUBSTITUTED TETRAHYDROPYRANS AND METHOD OF USE
Compounds of formula (I) ##STR00001## and pharmaceutically acceptable salts or radiolabelled forms thereof, wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5,...
2016/0122330 PIPERIDINYL BENZOIMIDAZOLE DERIVATIVES AS MPGE-1 INHIBITORS
The compounds (R)-1-(5-chloro-6-methyl-1-(6-(trifluoromethyl)pyridin-2-yl)-1H-benzo[d]i- midazol-2-yl)-N-(tetrahydrofuran-3-yl)piperidine-4-carboxamide and ...
2016/0122329 CRYSTALLINE FORMS OF AFATINIB DI-MALEATE
The present disclosure encompasses crystalline forms of Afatininb di-maleate and methods of their use.
2016/0122328 METHOD FOR PRODUCING AZOLE DERIVATIVE
In the present invention, a compound (I) is reacted with a base selected from the group consisting of a metal alkoxide, a metal hydride compound, an alkali...
2016/0122327 STROBILURIN TYPE COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI
The present invention relates to novel strobilurine type compounds I, processes for preparing these compounds, a use of compounds of the formula I and/or their...
2016/0122326 TRIAZOLE COMPOUNDS AND THEIR USE AS GAMMA SECRETASE MODULATORS
The present invention relates to compounds of formula (I) and pharmaceutically acceptable salts thereof. The invention also relates to pharmaceutical...
2016/0122325 Hydroxyalkyl-substituted phenyltriazole derivatives and uses thereof
The present invention relates to novel 5-(hydroxyalkyl)-1-phenyl-1,2,4-triazole derivatives, to processes for the preparation of such compounds, to...
2016/0122324 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS
The invention provides a novel class of compounds, pharmaceutical compositions comprising such compounds and methods of using such compounds to treat or...
2016/0122323 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7)
The present invention provides novel compounds of Formula (I), and pharmaceutically acceptable salts, solvates, hydrates, polymorphs, co-crystals, tautomers,...
2016/0122322 AZETIDINYLOXYPHENYLPYRROLIDINE COMPOUNDS
The invention provides certain azetidinyloxyphenylpyrrolidine compounds, particularly compounds of formula I wherein R is hydrogen or methyl, and ...
2016/0122321 Carboxamide Compounds and Methods for Using the Same
Disclosed are carboxamide compounds, as well as pharmaceutical compositions and methods of use. One embodiment is a compound having the structure ...
2016/0122320 USEFUL COMBINATIONS OF MONOBACTAM ANTIBIOTICS WITH BETA-LACTAMASE INHIBITORS
A pharmaceutical composition, comprising a combination of an antibiotically active compound of the formula (I): with a .beta.-lactamase inhibitor of one of the...
2016/0122319 CYCLIC AMINOMETHYL PYRIMIDINE DERIVATIVE
The present invention provides a cyclic aminomethyl pyrimidine derivative and a pharmaceutically acceptable salt thereof with high selectivity for dopamine...
2016/0122318 ISOINDOLINE INHIBITORS OF ROR-GAMMA
Provided are novel compounds of Formula (I): ##STR00001## pharmaceutically acceptable salts thereof, and pharmaceutical compositions thereof, which are useful in...
2016/0122317 1-SULFONYL PIPERIDINE DERIVATIVES AS MODULATORS OF PROKINETICIN RECEPTORS
##STR00001## The present invention provides compounds of formula (I) and pharmaceutically acceptable salts thereof in which m, n, W, X, Y, Z, R.sup.1,...
2016/0122316 SERINE/THREONINE KINASE INHIBITORS
Compounds of Formula I or a stereoisomer, tautomer, prodrug or pharmaceutically acceptable salt thereof are provided, which are useful for the treatment of...
2016/0122315 CRYSTALLINE IMATINIB MESYLATE PROCESS
The present invention relates to a process for preparation of crystalline non-needle shaped Form-SA of Imatinib mesylate (I). ##STR00001## The invention also...
2016/0122314 HISTONE DEMETHYLASE INHIBITORS
The present invention relates generally to compositions and methods for treating cancer and neoplastic diseases. Provided herein are substituted ...
2016/0122313 COMPOSITIONS AND METHODS FOR THE TREATMENT OF DIABETES
The invention relates to the compounds of formula I or its pharmaceutical acceptable salts, as well as polymorphs, solvates, enantiomers, stereoisomers and...
2016/0122312 ANTI-VIRAL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF
Disclosed herein are compounds, pharmaceutical compositions, and methods for the treatment of viral infection, including RNA viral infection, as well as...
2016/0122311 SYNTHESIS OF COUMALIC ACID
A method to prepare coumalic acid comprising (a) heating a solution in dichloroethane of malic acid and sulfuric acid or a solution in dichloroethane of malic...
2016/0122310 PROCESS FOR THE MANUFACTURE OF EPOXY-MONOMERS AND EPOXIDES
A process for manufacturing epoxy monomers and/or epoxides in high yields and useful quality and chemical stability by dehydrochlorination of the corresponding...
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