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CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS
Chemical entities that are novel compounds, pharmaceutical compositions and methods of treatment of cancer are described.
STEROIDS HAVING INCREASED WATER SOLUBILITY AND RESISTANCE AGAINST
METABOLISM AND METHODS FOR THEIR PRODUCTION
Steroid compounds having increased resistance against metabolism and increased water solubility are disclosed, together with methods for their production....
NOVEL REAGENTS FOR UNIVERSAL SITE-SPECIFIC LABELING AND MODIFICATIONS OF
The present invention discloses a method of harnessing versatile phosphoramidation reactions to regioselectively incorporate alkynyl/azido groups into...
NICOTINIC ACID RIBOSIDE OR NICOTINAMIDE RIBOSIDE COMPOSITIONS, REDUCED
DERIVATIVES THEREOF, AND THE USE THEREOF...
Derivatives of nicotinic acid riboside (NAR), nicotinamide riboside (NR), and reduced NAR and NR, including ...
PRODUCTION OF RHAMNOLIPID COMPOSITIONS
Provided are organic solvent free methods for obtaining compositions comprising one or more rhamnolipids as well as compositions obtainable from said methods.
Partially Crystalline Glucamide Compositions And Method For Preparing Same
The invention relates to a partially crystalline N-alkyl-N-acylglucamine composition comprising at least two different acylglucamines with acyl groups selected...
PRODUCTION OF RENEWABLE FINE CHEMICALS AND LIQUID FUELS
Described herein is a process for conversion and upgrading of biomass to products. The process involves converting the biomass to primary lignin-derivatives...
RUTHENIUM COMPOUND, MATERIAL FOR THIN FILM FORMATION, AND PROCESS FOR THIN
Disclosed is a ruthenium compound useful as a precursor in chemical vapor growth, particularly ALD. The compound has good reactivity with a reactive gas, a...
OSMIUM (II) ARENE AZO ANTI-CANCER COMPLEXES
The present invention relates to the use of certain osmium containing complexes such as cytotoxic agents particularly for the treatment of cancer. There is...
GENERAL CATALYST FOR C-H FUNCTIONALIZATION
The invention provides novel manganese catalysts such as [Mn(.sup.tBuPc)], which are general for the amination of all types of C(sp.sup.3)-H bonds (aliphatic,...
PURIFIED PHOSPHATIDYLCHOLINE PRODUCT MADE BY A PROCESS EMPLOYING MAGNETIC
A process for separation and purification of phosphatides, especially phosphatidylcholine, from vegetable lecithins, comprising deoiling with acetone,...
METHOD FOR THE PURIFICATION OF LECITHIN
The present invention relates to a method for the purification of lecithin, comprising the steps of (a) mixing lecithin with active carbon to form a...
PREPARATION OF TITANIUM CATECHOLATE COMPLEXES IN AQUEOUS SOLUTION USING
TITANIUM TETRACHLORIDE OR TITANIUM...
Titanium coordination complexes, particularly titanium catecholate complexes, can be attractive active materials for use in flow batteries. However, such...
Process to Prepare Aluminoxanes by Reaction of Alkylaluminium With Allylic
The present invention relates to a process to prepare alkylaluminoxanes by reaction of alkylaluminium with a substituted allylic alcohol of the formula wherein...
HIGHLY FLUORESCENT PYRROLE-BF2 CHROMOPHORES
Fluorescent chromophores nicknamed BOPHY are provided. The chromophores may be readily synthesized in two steps from readily available reagents via the...
SINGLE MOLECULE AND ORGANIC SOLAR CELL COMPRISING SAME
The present specification provides a single molecule and an organic solar cell including the same.
TRICYCLIC PIPERIDINE COMPOUNDS
The present invention relates to compounds of the formula (I) ##STR00001## wherein R, R.sup.1a, R.sup.1b, R.sup.2, R.sup.3, and X are as described in the...
SPIROCYCLIC DIHYDRO-THIAZINE AND DIHYDRO-OXAZINE BACE INHIBITORS, AND
COMPOSITIONS AND USES THEREOF
Compounds are provided having a structure according to Formula (I): wherein A.sub.1, A.sub.2, A.sub.3, Y, R.sub.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6,...
PRO-DRUGS OF NSAIAS WITH VERY HIGH SKIN AND MEMBRANES PENETRATION RATES
AND THEIR NEW MEDICINAL USES
The novel positively charged pro-drugs of NSAIAs in the general formulas (1, 2a, 2b, 2c, or 2d) "Structure 1, 2a, 2b, 2c, or 2d" were designed and synthesized....
BENZO-THIAZOLO-IMIDAZOLE COMPOUNDS AND USES THEREOF
The present invention relates to benzo-thiazolo-imidazole compounds and their uses. Moreover, the present invention relates to pharmaceutical compositions...
DGAT1 Inhibitor and Preparation Method and Use Thereof
The present invention discloses a novel DGAT1 inhibitor, especially the compound of formula (I) or a pharmaceutically acceptable salt thereof, preparation and...
PYRANOCHROMENYL PHENOL DERIVATIVE, AND PHARMACEUTICAL COMPOSITION FOR
TREATING METABOLIC SYNDROME OR...
Provided are a pyranochromenyl phenol derivative, a pharmaceutically acceptable salt thereof, or a solvate thereof. Also provided is a pharmaceutical...
DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE
This invention is directed to compounds of formula (I): ##STR00001## where r, q, R, R.sup.2, R.sup.3, R.sup.4, R.sup.5a, R.sup.5b, R.sup.5c, R.sup.6a, R.sup.6b,...
Heteroaryl Substituted Pyrrolo[2,3-B] Pyridines And Pyrrolo[2,3-B]
Pyrimidines As Janus Kinase Inhibitors
The present invention provides heteroaryl substituted pyrrolo[2,3-b]pyridines and heteroaryl substituted pyrrolo[2,3-b]pyrimidines that modulate the activity...
PYRAZOLOPYRIDAZINES AND METHODS FOR TREATING RETINAL-DEGENERATIVE DISEASES
AND HEARING LOSS ASSOCIATED WITH...
Compounds, compositions and methods for the treatment of retinal degenerative diseases, such as retinitis pigmentosa, Leber's congenital Amaurosis, Syndromic...
RESPIRATORY SYNCYTIAL VIRUS INHIBITORS
Compounds of Formula (I), wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4 and n are defined herein, are useful as inhibitors of RSV. ##STR00001##
Heterocyclic Compounds and Methods of Use
The present application discloses compounds that are inhibitors of Btk, compounds that are inhibitors of PI3K.delta., and compounds that are dual inhibitors of...
METHOD OF STABILIZING RIBOFLAVIN
A method of stabilizing riboflavin by affixing the riboflavin to at least one substrate for the riboflavin by covalent bonding, hydrogen bonding, Van der Waals...
5'-NUCLEOTIDASE INHIBITORS AND THERAPEUTIC USES THEREOF
The subject matter of the present invention is compounds which have a 6-aminopurine backbone corresponding to formula (I): in which R.sub.1, R.sub.2, R.sub.3,...
PROCESS FOR THE PREPARATION OF DIPEPTIDYLPEPTIDASE INHIBITORS
The present invention provides a process for the preparation of linagliptin, a compound of Formula I, the process comprising deprotecting a compound of Formula...
CRYSTALLINE FORMS OF DIAZABICYCLOOCTANE DERIVATIVE AND PRODUCTION PROCESS
A crystalline form of a diazabicyclooctane derivative represented by the following Formula (VII), and processes for producing the same: ##STR00001##
SUBSTITUTED PIPERIDIN-4-AMINO-TYPE COMPOUNDS AND USES THEREOF
The disclosure relates to Substituted Piperidin-4-amino-Type Compounds of Formula (I) and pharmaceutically acceptable salts and solvates thereof wherein...
COMPOUNDS AND METHODS FOR THE ENHANCED DEGRADATION OF TARGETED PROTEINS
The present invention relates to bifunctional compounds, which find utility as modulators of targeted ubiquitination, especially inhibitors of a variety of...
PESTICIDALLY ACTIVE BICYCLIC HETEROCYCLES WITH SULPHUR CONTAINING
Compounds of the formula (I), and the agrochemically acceptable salts and N-oxides of those compounds, including all stereoisomers and tautomeric forms, and...
SUBSTITUTED OXOPYRIDINE DERIVATIVES
The invention relates to substituted oxopyridine derivatives and to processes for their preparation, and also to their use for preparing medicaments for the...
CRYSTAL FORM OF (R)-PRAZIQUANTEL AND PREPARATION METHOD AND APPLICATION
The present invention relates to a crystal form of (R)-praziquantel and a preparation method and uses thereof. The X-ray diffraction pattern (CuK.alpha....
SUBSTITUTED DIHYDROPYRIDO[3,4-B]PYRAZINONES AS DUAL INHIBITORS OF BET
PROTEINS AND POLO-LIKE KINASES
The present invention relates to substituted dihydropyrido[3,4-b]pyrazinones as dual inhibitors of BET proteins, in particular BRD4 proteins, and Polo-like...
ACYCLIC CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS
The instant invention provides compounds of formula I which are JAK inhibitors, and as such are useful for the treatment of JAK-mediated diseases such as...
N-(2-CYANO HETEROCYCLYL) PYRAZOLO PYRIDONES AS JANUS KINASE INHIBITORS
Provided are compounds of Formula I, a JAK inhibitor, and use thereof for the treatment of JAK-mediated diseases by the application. ##STR00001##
GEMINALLY SUBSTITUTED CYANOETHYLPYRAZOLO PYRIDONES AS JANUS KINASE
The instant invention provides compounds of Formula (I) which are JAK inhibitors, and as such are useful for the treatment of JAK-mediated diseases such as...
KETO-IMIDAZOPYRIDINE DERIVATIVES AS RORc MODULATORS
Compounds of the formula I or II: ##STR00001## or pharmaceutically acceptable salts thereof, wherein R.sup.1 is a group of formula (a), (b), (c); (d) or (e): ...
Compounds of formula (I) and pharmaceutically acceptable salts thereof are provided. The compounds are useful as agents in the treatment of diseases and...
PROCESS FOR THE PREPARATION OF BENZOHETERO [1,3] - DIAZOLE COMPOUNDS
DISUBSTITUTED WITH HETEOARYL GROUPS
Process for the preparation of a benzohetero[1,3]diazole compound disubstituted with heteroaryl groups which comprises reacting at least one...
NOVEL 3-INDOL SUBSTITUTED DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND
METHODS FOR USE
A compound of Formula I is provided: ##STR00001## or pharmaceutically acceptable enantiomers, salts or solvates thereof. The invention further relates to the use...
POLYMORPHIC FORMS OF SUVOROXANT
Present invention relates to crystalline form of suvorexant, amorphous form of suvorexant, amorphous solid dispersion of suvorexant, processes for their...
The present invention relates to compounds of formula ##STR00001## wherein R.sup.1/R.sup.2 are hydrogen, lower alkyl, lower alkoxy, lower alkyl substituted by...
HETEROCYCLIC SULFONAMIDES, USES AND PHARMACEUTICAL COMPOSITIONS THEREOF
The invention is directed to a class of compounds, including the pharmaceutically acceptable salts of the compounds, having the structure of formula I: ...
METHODS FOR PREPARING BREXPIPRAZOLE, KEY INTERMEDIATES THEREOF AND SALTS
The present invention relates to the methods for preparing brexpiprazole, the analogs, key intermediates, and salts thereof, specifically, the present...
FORMATION OF MACROMOLECULES USING ITERATIVE GROWTH AND RELATED COMPOUNDS
In some embodiments, macromolecules and related methods are provided. In some embodiments, an iterative growth process may be used to form a macromolecule...
TETRAZOLINONE COMPOUND AND USE THEREOF
A tetrazolinone compound represented by formula (1) ##STR00001## wherein E represents the following group E16; ##STR00002## Y represents --O--CH.sub.2--; Q...