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Patent # Description
2018/0186812 PROCESS FOR PREPARING CARBAMOYLPYRIDONE DERIVATIVES ANDINTERMEDIATES
The present invention relates to the preparation of carbamoylpyridone derivatives such as the compound of formula (VIIIa): ##STR00001##
2018/0186811 Process for preparing carbamoylpyridone derivatives and intermediates
The present invention relates to the preparation of carbamoylpyridone derivatives such as the compound of formula (VIIIa): ##STR00001##
2018/0186810 STEREOCHEMICALLY DEFINED POLYPROPIONATES AND METHODS FOR MAKING AND USING THE SAME
The present invention relates to stereochemically defined polypropionates and methods for preparing and using the same. The stereochemically defined...
2018/0186809 PROCESS FOR PRODUCTION OF A SPIROGLYCOL
Disclosed is a process for production of a spiroglycol by subjecting pentaerythritol to reaction in water with hydroxypivaldehyde in presence of a...
2018/0186808 NARGENICIN COMPOUNDS AND USES THEREOF AS ANTIBACTERIAL AGENTS
The present invention relates to novel nargenicin related compounds which can inhibit DnaE and have antibacterial, particularly antimycobacterial activity...
2018/0186807 COMPOUNDS AND USES THEREOF FOR THE MODULATION OF HEMOGLOBIN
Provide herein are compounds and pharmaceutical compositions suitable as modulators of hemoglobin, methods and intermediates for their preparation, and methods...
2018/0186806 ANTIVIRAL COMPOUNDS
The disclosure is related to anti-viral compounds, compositions containing such compounds, and therapeutic methods that include the administration of such...
2018/0186805 PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-alpha]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2- ...
The present disclosure relates to processes for preparing (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]pyrazin-8-yl)-N-(2,2,2-- ...
2018/0186804 METHOD FOR PREPARING SPIRO QUATERNARY AMMONIUM SALT
The present invention relates to a method for preparing a spiro quaternary ammonium salt comprising reacting a cyclic secondary amine with a dihaloalkane in...
2018/0186803 SHORT-ACTING BENZODIAZEPINE SALTS AND THEIR POLYMORPHIC FORMS
The invention relates to besylate salts of the compound of formula (I): ##STR00001## Methods of preparing the salts, and their use as medicaments, in particular...
2018/0186802 COMPOUNDS AND COMPOSITIONS AS TOLL-LIKE RECEPTOR 7 AGONISTS
The invention provides compounds of Formula (I), immunogenic compositions and pharmaceutical compositions comprising such compounds and methods of using such...
2018/0186801 SUBSTITUTED BICYCLIC AZA-HETEROCYCLES AND ANALOGUES AS SIRTUIN MODULATORS
Provided herein are novel substituted bicyclic aza-heterocycle sirtuin-modulating compounds and methods of use thereof. The sirtuin-modulating compounds may be...
2018/0186800 BRK INHIBITORY COMPOUND
The present invention relates to a compound represented by general formula (I) (wherein, all symbols represent the same meanings as the symbols set forth in...
2018/0186799 HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS
Disclosed are compounds of Formula (I) or salts thereof, wherein HET is a heteroaryl selected from pyrrolo[2,3-b]pyridinyl, pyrrolo[2,3 d]pyrimidinyl,...
2018/0186798 PRMT5 INHIBITORS AND USES THEREOF
Described herein are compounds of Formula (I), pharmaceutically acceptable salts thereof, and pharmaceutical compositions thereof. Compounds of the present...
2018/0186797 5-HT2C RECEPTOR AGONISTS AND COMPOSITIONS AND METHODS OF USE
Provided in some embodiments are compounds herein. Also provided in some embodiments are methods for weight management, inducing satiety, and decreasing food...
2018/0186796 COMPOUNDS AND USES THEREOF
The present invention refers to 4-amino-substituted pyrazolo[3,4-d]pyrimidine and pyrrolo[2,3-d]pyrimidine derivatives of formula I and IV able to target the...
2018/0186795 PYRIMIDINONES AS FACTOR XIA INHIBITORS
The present invention provides compounds of Formula (I): ##STR00001## or stereoisomers, tautomers, or pharmaceutically acceptable salts thereof, wherein all the...
2018/0186794 IMIDAZOPYRROLOQUINOLINE SALT, METHOD FOR PRODUCING THE SAME, MEDICAMENT, COSMETIC, AND FOOD
There is provided a production method for the purpose of improving the solubility of an arginine-residue imidazopyrroloquinoline in water and making the purity...
2018/0186793 P2X3 AND/OR P2X2/3 COMPOUNDS AND METHODS
The present application provides novel compounds and methods for preparing and using these compounds. In one embodiment, the compounds are of the structure of...
2018/0186792 HETEROBIFUNCTIONAL LINKERS WITH POLYETHYLENE GLYCOL SEGMENTS AND IMMUNE RESPONSE MODIFIER CONJUGATES MADE THEREFROM
Conjugates of an immune response modifier, a linker, and an antigen are disclosed. The linker is represented by formula: ##STR00001## wherein A is CH or N, p is...
2018/0186791 SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORS
Provided herein are compounds of the General Formula I: ##STR00001## and stereoisomers and pharmaceutically acceptable salts or solvates thereof, in which A, B,...
2018/0186790 SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORS
Provided herein are compounds of the General Formula I: ##STR00001## and stereoisomers and pharmaceutically acceptable salts or solvates thereof, in which A, B,...
2018/0186789 PYRAZOLOPYRIDINE DERIVATIVES AND THEIR USE IN THERAPY
The present invention relates to pyrazolopyridine derivatives, which are useful as medicaments, pharmaceutical compositions comprising one or more of the...
2018/0186788 CRYSTALLINE FORM OF FUSED PYRIDINE DERIVATIVE'S MALEATE AND USES THEREOF
The compound of Formula I, the crystalline form thereof, and methods of preparing and using them are provided. ##STR00001##
2018/0186787 PHARMACEUTICAL COMPOUND
Provided is a tryptophan-2,3-dioxygenase (TDO) and/or indoleamine-2,3-dioxygenase (IDO) inhibitor compound for use in medicine, which compound comprises the...
2018/0186786 A CASEIN KINASE 1 DELTA INHIBITOR
The present invention provides 2-Methyl-amino-3-[(4-fluorophenyl)carbonyl]indolizine-1-carboxamide of formula (I) or a pharmaceutically acceptable salt...
2018/0186785 Proteolysis Targeting Chimera Compounds and Methods of Preparing and Using Same
The present invention includes novel compounds and methods for preventing or treating diseases associated with and/or caused by overexpression and/or...
2018/0186784 CRYSTALLINE FORMS OF N-(2-CHLORO-6-METHY]PHENVN-2-[F6-[4-(2-HVDROXVETHVL)-L-PIPERAZIN-VIL-2-ME- ...
The present invention relates to crystalline 1,2-Propanediol solvate of N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1-piperazinyl]-2-me- ...
2018/0186783 INHIBITORS OF PROTEIN KINASES
The present invention is directed to compounds of formula I-II and pharmaceutically acceptable tautomers, salts, or stereoisomers thereof which are inhibitors...
2018/0186782 AMIDE COMPOUNDS FOR TREATMENT OF IMMUNE AND INFLAMMATORY DISORDERS
Compounds, methods of use, and processes for making inhibitors of complement Factor D are provided comprising Formula I, I'' and I''' or a pharmaceutically...
2018/0186781 BICYCLO[1.1.1]PENTANE INHIBITORS OF DUAL LEUCINE ZIPPER (DLK) KINASE FOR THE TREATMENT OF DISEASE
Disclosed herein are compounds which inhibit the kinase activity of dual leucine zipper (DLK) kinase (MAP3K12), pharmaceutical compositions, and methods of...
2018/0186780 METHODS TO TREAT LYMPHOPLASMACYTIC LYMPHOMA
The present invention provides compounds of any one of Formulae (I) to (V) (e.g., compounds of any one of Formulae (I-1) to (I-9)), and methods for treating...
2018/0186779 G PROTEIN-COUPLED RECEPTOR KINASE INHIBITORS AND METHODS FOR USE OF THE SAME
Disclosed herein are novel GRK inhibitors and methods for their use in treating or preventing heart disease, such as cardiac failure, cardiac hypertrophy, and...
2018/0186778 HETEROARYL-1,2,4-TRIAZOLE AND HETEROARYL-TETRAZOLE COMPOUNDS FOR CONTROLLING ECTOPARASITES
The present invention provides compounds of the formula: (I) wherein: X is O or S; Q.sup.1 and Q.sup.2 are independently CR.sup.5 or N, provided at least one...
2018/0186777 SULFONAMIDE COMPOUNDS AS VOLTAGE-GATED SODIUM CHANNEL MODULATORS
The present invention relates to sulfonamide compounds Formula (I) wherein the substituents are as described herein, and their use in a medicine for the...
2018/0186776 HESPERETIN AZA-CINNAMIC ACID DERIVATIVES WITH ANTI-TUMOR ACTIVITIES AND A METHOD OF PREPARING THE SAME
A hesperetin aza-cinnamic acid derivative has the following formula (I): ##STR00001## R.sub.1 is H or alkyl, and R.sub.2 and R.sub.2 are independently H, alkyl,...
2018/0186775 QUINOXALINE DERIVATIVES USEFUL AS FGFR KINASE MODULATORS
The invention relates to new quinoxaline derivative compounds, to pharmaceutical compositions comprising said compounds, to processes for the preparation of...
2018/0186774 NOVEL ANNELATED BENZAMIDES
The present invention relates to compounds of formula (I) ##STR00001## wherein R.sup.1, R.sup.2, and Z.sup.- have one of the meanings as indicated in the...
2018/0186773 METALLOENZYME INHIBITOR COMPOUNDS
Provided are compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.
2018/0186772 6-(5-HYDROXY-1H-PYRAZOL-1-YL)NICOTINAMIDE INHIBITORS OF PHD
The present invention provides compounds of the formula: ##STR00001## which are useful as inhibitors of PHD, pharmaceutical compositions thereof, methods for...
2018/0186771 INDOLIZINE COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
Compounds of formula (I) wherein Ra, Rb, Rc, Rd, T, R3, R4, R5, X, Y and Het are as defined in the description. ##STR00001## Medicinal products containing the...
2018/0186770 COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF SHP2
The present invention relates to compounds of formula I: ##STR00001## in which Y.sub.1, Y.sub.2, Y.sub.3, R.sub.1, R.sub.2, R.sub.4a, R.sub.5b, R.sub.5a,...
2018/0186769 6-AMINO-5-FLUORO-5-(FLUOROMETHYL)-2,3,4,5-TETRAHYDROPYRIDIN-2-YL-PHENYL-5-- (METHOXY-D3)-PYRAZINE-2-CARBOXAMIDES...
The invention provides amidine compounds of Formula I ##STR00001## for the treatment of neurodegenerative or cognitive diseases, including Alzheimer's Disease.
2018/0186768 Antibacterial Compounds
The present invention relates to the following compounds ##STR00001## wherein the integers are as defined in the description, and where the compounds may be...
2018/0186767 ANTIPROLIFERATIVE COMPOUNDS, AND THEIR PHARMACEUTICAL COMPOSITIONS AND USES
Compounds of formula A-I and B-I, compositions comprising the compounds, methods of making the compounds and methods of their uses are disclosed.
2018/0186766 PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS
This application relates to efficient and economical synthetic chemical processes for the preparation of pesticidal thioethers and pesticidal sulfoxides....
2018/0186765 PROCESSES FOR THE PREPARATION OF PESTICIDAL COMPOUNDS
This application relates to efficient and economical synthetic chemical processes for the preparation of pesticidal thioethers and pesticidal sulfoxides....
2018/0186764 ORGANIC COMPOUND, ORGANIC OPTOELECTRIC DIODE, AND DISPLAY DEVICE
The present invention relates to an organic compound represented by Chemical Formula 1, an organic optoelectronic diode, and a display device.
2018/0186763 Method for Producing Fluorine-Containing Cyclopropane Carboxylic Acid Compound
The present invention provides an industrially applicable method for production of a fluorine-containing cyclopropane carboxylic acid compound useful as an...
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