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Patent # Description
US-9,353,098 Polymorphs and salts
The present invention is directed to novel polymorphs and salts of a compound which is an inhibitor of kinase activity.
US-9,353,097 Solid state forms of a quinazoline derivative and its use as a BRAF inhibitor
This application relates to various salts and solid state forms of Compound (I). This application also relates to pharmaceutical compositions and therapeutic...
US-9,353,096 Substituted phenylcarbamate compounds
The invention is concerned with the compounds of formula (I): ##STR00001## and pharmaceutically acceptable salts thereof, wherein Y, R1, R2 and R3 are defined...
US-9,353,095 Crystalline form A of 1,5-dimethyl-6-thioxo-3-(2,2,7-trifluoro-3-oxo-4-(prop-2-ynyl)-3,4-dihydr- ...
The present invention relates to a novel crystalline form A of 1,5-dimethyl-6-thioxo-3-(2,2,7-trifluoro-3-oxo-4-(prop-2-ynyl)-3,4-dihydr- ...
US-9,353,094 Substituted quinoxalines as kinase inhibitors
Disclosed herein are compounds of formula (I) and methods of inhibiting IKK.beta. and the NF-.kappa.B signaling and mTOR pathways. ##STR00001##
US-9,353,093 Indole-1-carboxamides as kinase inhibitors
This invention is directed to a compound of Formula I ##STR00001## or a pharmaceutically acceptable salt thereof, wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4,...
US-9,353,092 Synthesis and use of croconaine compounds
The present disclosure provides compositions and methods for the synthesis and use of croconaine compounds. The disclosed compounds are easily prepared from...
US-9,353,091 Antiviral compounds and uses thereof
This invention relates to: (a) compounds and salts thereof that, inter alia, inhibit HCV; (b) intermediates useful for the preparation of such compounds and...
US-9,353,090 Heterocyclic carboxylic acids as activators of soluble guanylate cyclase
The present invention relates to compounds of formula I: ##STR00001## and pharmaceutically acceptable salts thereof, wherein R.sup.1, R.sup.2, R.sup.3,...
US-9,353,089 Compositions and methods for the treatment of malaria
The present invention provides aminohydantoin anti-malarial agents. In some embodiments, these agents have the property of functions of targeting malarial...
US-9,353,088 Crystalline pharmaceutical and methods of preparation and use thereof
Novel crystalline polymorphic forms, Forms A, B, C, D, and E of a compound of Formula I, which has been found to be a potent inhibitor of LFA-1, are disclosed....
US-9,353,087 Inhibitors of Bruton's tyrosine kinase
The present invention provides a compound, solid forms, and compositions thereof, which are useful as inhibitors of Bruton's tyrosine kinase and which exhibit...
US-9,353,086 CXCR4 receptor antagonists
Disclosed are compounds that are antagonists of the CXCR4 receptor.
US-9,353,085 Compound for organic electroluminescent device and organic electroluminescent devices using the same
The present invention provides a compound of formula (I) for an organic electroluminescent device: ##STR00001## wherein X.sub.1, X.sub.2, X.sub.3, Y,...
US-9,353,084 2-amino 3,5,5-trifluoro-3,4,5,6-tetrahydropyridines as BACE1 inhibitors for treatment of Alzheimer's disease
The present invention is directed to novel inhibitors of the BACE1 enzyme. Separate aspects of the invention are directed to pharmaceutical compositions...
US-9,353,083 Oxazetidine derivatives, process for preparing them and use in human medicine and in cosmetics
Methods for treating hypopigmentary pathologies and photosensitive dermatoses are described. Also described, are compounds that are agonists of the MCIR...
US-9,353,082 Pharmaceutical compounds
The invention relates to compounds and compositions for inhibiting the enzyme fatty acid amide hydrolase (FAAH), the use of the compounds in therapy and, in...
US-9,353,081 Bicyclic dihydroquinoline-2-one derivatives
The invention provides novel compounds having the general formula (I) ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, R.sup.7,...
US-9,353,080 Polymorphic forms of 3-(4-amino-1-oxo-1,3 dihydro-isoindol-2-yl)-piperidine-2,6-dione
Polymorphic forms of 3-(4-amino-1-oxo-1,3 dihydro-isoindol-2-yl)-piperidine-2,6-dione are disclosed. Compositions comprising the polymorphic forms, methods of...
US-9,353,079 Solid forms of an alpha, omega di-substituted dihydroxy cyclopentyl compound and methods for the preparation...
Provided herein are multiple solid forms of a defined .alpha.,{acute over (.omega.)}-disubstituted dihydroxy cyclopentyl compound, and methods for the...
US-9,353,078 Amino, amido and heterocyclic compounds as modulators of rage activity and uses thereof
Amino, amido, and heterocyclic compounds are disclosed. The compounds may be prepared as pharmaceutical compositions, and may be used for the prevention and...
US-9,353,077 Organocatalytic process for asymmetric synthesis of decanolides
The present invention discloses organocatalytic process for asymmetric synthesis of highly enantioselective decanolide compounds in high yield with >99% ee....
US-9,353,076 Crystal form of cabazitaxel and preparation method thereof
The present invention relates to the field of medical chemistry, and discloses a preparing method for three crystal forms of cabazitaxel, that is, crystalline...
US-9,353,075 Disubstituted beta-lactones as inhibitors of N-acylethanolamine acid amidase (NAAA)
The present invention provides compounds and pharmaceutical compositions for inhibiting N-acylethanolamine acid amidase (NAAA). Inhibition of NAAA is...
US-9,353,074 Thermally integrated process for the production of ethylene oxide from a flow of ethanol
Process for dehydrating an ethanol feed to ethylene then oxidating the ethanol to ethylene oxide, comprising vaporizing the feed and a flow of diluting water...
US-9,353,073 Vortioxetine manufacturing process
A process for the manufacture of vortioxetine is provided in which a compound of formula I, formula I is reacted with optionally substituted piperazine and...
US-9,353,072 Antimicrobial substituted thiazoles and methods of use
Disclosed are compositions having activity against MRSA and/or VRSA, and methods of using the compositions to treat microbial infections.
US-9,353,071 Method for manufacturing isothiazole compound
An industrially preferred process for producing an isothiazole compound, particularly 3,4-dichloro-5-cyanoisothiazole, provides a safer industrial production...
US-9,353,070 Carbamat-benzoxazinones
The present invention relates to carbamat-benzoxazinones of formula (I), ##STR00001## wherein the variables are defined according to the description, as well...
US-9,353,069 Super-oxide dismutase mimetics
The present invention relates to compounds which are effective as catalysts for dismutating superoxide and, more particularly, the manganese or iron complexes...
US-9,353,068 3-heteroaroylamino-propionic acid derivatives and their use as pharmaceuticals
The present invention relates to compounds of the formula I, ##STR00001## wherein Ht, G, R.sup.10, R.sup.30, R.sup.40, R.sup.50 and R.sup.60 have the meanings...
US-9,353,067 Heterocyclic compounds and uses thereof in the treatment of sexual disorders
Biologically active compounds, which are useful for treating a sexual disorder, are provided herein. Further provided are pharmaceutical compositions formulated...
US-9,353,066 Substituted phenyl-Spleen Tyrosine Kinase (Syk) inhibitors
The invention provides certain substituted phenyl compounds of the Formula (I) or pharmaceutically acceptable salts thereof, wherein R.sup.1, R.sup.2, R.sup.3,...
US-9,353,065 Heterocyclic bridged biphenyls
The present invention relates to compounds of the formula (I), a process for their preparation and their use in organic light emitting diodes (OLEDs),...
US-9,353,064 Processes useful for the preparation of ...
The present invention is directed to processes and intermediates useful for the preparation of ...
US-9,353,063 Opsin-binding ligands, compositions and methods of use
Compounds are disclosed that are useful for treating ophthalmic conditions caused by or related to production of toxic visual cycle products that accumulate in...
US-9,353,062 Substituted quinolines as bruton's tyrosine kinases inhibitors
The present invention is directed to novel quinolines, their derivatives, pharmaceutically acceptable salts, solvates and hydrates thereof. The compounds and...
US-9,353,061 3,5,N-trihydroxy-alkanamide and derivatives: method for making same and use thereof
The present invention provides novel compounds of Formula (I), and pharmaceutically compositions thereof. Compounds of Formula (I) are inhibitors of histone...
US-9,353,060 Process for the preparation of 3-hydroxypicolinic acids
4,6-Dibromo-3-hydroxypicolinate esters are prepared from furan-2-yl aminoacetates in one chemical step by use of a bromination-rearrangement reaction.
US-9,353,059 Donepezil pamoate, method of preparation and use thereof
The composition containing a pamoate salt of donepezil, the method of preparation and the use thereof are disclosed.
US-9,353,058 Anti-parasitic methods and compositions utilizing diindolylmethane-related indoles
The present invention includes methods and compositions for the treatment and prevention of protozoal parasitic infections utilizing Diindolylmethane-related...
US-9,353,057 Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
Methods for synthesis of 1-(acyloxy)-alkyl carbamates, particularly, the synthesis of 1-(acyloxy)-alkyl carbamate prodrugs of primary or secondary ...
US-9,353,056 Zwitterionic reagents
Zwitterion-containing compounds for the modification of hydrophobic molecules to improve their solubility and/or to lower their non-specific binding as...
US-9,353,055 Method for the purification of prostaglandins
The present invention provides a method for the purification of a prostaglandin by supercritical fluid chromatography, said method comprising the use of a...
US-9,353,054 Hydrotreating catalyst sulphiding agent and its use for in situ and ex situ presulphidation
The present invention relates to a sulphiding agent for a hydrotreating catalyst which makes possible faster sulphiding of the catalyst but which also makes...
US-9,353,053 Thiolation method for modifying carbon nanotubes
A thiolation method for modifying carbon nanotubes includes steps as follows. A carboxylation step is provided, wherein the carbon nanotubes are reacted with an...
US-9,353,052 Fluorinated oligomers having pendant bromine-containing moieties
Described herein is an oligomer having a pendant bromine-containing moiety according to formula II and/or formula III; and combinations thereof; wherein...
US-9,353,051 Antiviral drugs for treatment or prevention of dengue infection
Compounds, methods and pharmaceutical compositions for treating viral infections, by administering certain compounds in therapeutically effective amounts are...
US-9,353,050 Process for preparation of isosulfan blue
A process for the preparation of isosulfan blue (Active Pharmaceutical Ingredient) is provided. A process is also provided for preparation of the intermediate,...
US-9,353,049 Preparation method for rivastigmine, intermediates thereof, and preparation method for said intermediates
The present invention provides a preparation method for (S)-3-(1-(dimethylamino)ethyl)phenyl ethyl(methyl)carbamate, preparation methods for intermediates ...
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