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Patent # Description
US-9,359,351 Cap/endo dual inhibitors and their use in the treatment, amelioration or prevention of a viral disease
The present invention relates to a compound having the general formula (V), optionally in the form of a pharmaceutically acceptable salt, solvate, polymorph,...
US-9,359,350 Ring-fused compound
The present invention relates to a compound that has URAT1 inhibitory action, and a URAT1 inhibitor, a blood uric acid level-reducing agent and a pharmaceutical...
US-9,359,349 Substituted quinazolines as kinase inhibitors
The present invention provides compounds of Formula I ##STR00001## that modulate PI3 kinase activity and methods of treatment of diseases and conditions...
US-9,359,348 Cyclopropyl imidazopyridine PDE10 inhibitors
The present invention is directed to substituted cyclopropyl imidazopyridine compounds which are useful as therapeutic agents for the treatment of central...
US-9,359,347 Inhibitors of Akt/PKB with anti-tumor activity
The subject invention concerns materials and methods for inhibiting the Akt/PKB pathway. In one embodiment, a compound of the invention inhibits kinase activity...
US-9,359,346 Benzamide derivative and use thereof
Disclosed are a novel benzamide derivative and pharmaceutical use thereof, and more particularly, a novel benzamide derivative having a structure of Formula 1...
US-9,359,345 Thiazole derivatives as inhibitors of Bruton's tyrosine kinase
This application discloses compounds according to generic Formula I: wherein all variables are defined as described herein, which inhibit Btk. The compounds...
US-9,359,344 Biaryl heterocycle substituted oxazolidinone antibacterial agents
The present invention relates to a biaryl heterocycle substituted oxazolidinone antibacterials shown by general formula (I), a pharmaceutically acceptable salt...
US-9,359,343 Fluorine atom-containing disulfide compound
A disulfide compound represented by formula (1): ##STR00001## (in formula (1), R.sub.1 and R.sub.2 each independently represent a hydrogen atom or an alkyl...
US-9,359,342 Protein disulfide isomerase inhibiting anticancer agents
Protein disulfide isomerase inhibitors according to formula I ##STR00001## are described, wherein R.sup.1 is an aryl or cycloalkyl group, R.sup.2 is selected...
US-9,359,341 Aldehyde derivative of substitute oxazolidinones
The present invention relates to the prodrug of 5-chloro-N-({(5S)-2-oxo-3-[4-(3-oxo-morpholin-4-yl)phenyl]-1,3-oxazolidin- -5-yl}methyl)thiophene-2-carboxamide,...
US-9,359,340 Hydroxylated and methoxylated pyrimidyl cyclopentanes as Akt protein kinase inhibitors
The present invention provides compounds, including resolved enantiomers, resolved diastereomers, solvates and pharmaceutically acceptable salts thereof,...
US-9,359,339 Glucagon receptor antagonist compounds, compositions containing such compounds and methods of use
Glucagon receptor antagonist compounds are disclosed. The compounds are useful for treating type 2 diabetes and related conditions. Pharmaceutical compositions...
US-9,359,338 Cyclopropanecarboxamido-substitute aromatic compounds as anti-tumor agents
Provided are cyclopropanecarboxamido-substituted aromatic compounds that inhibit protein kinases and their use in anti-tumor area. In particular, ...
US-9,359,337 Acetamide derivatives
The invention is concerned with a compound of formula (I) ##STR00001## and pharmaceutically acceptable salts thereof wherein R1 to R3, X and Y are as defined...
US-9,359,336 Heterocycle-substituted pyridyl benzothiophenes as kinase inhibitors
This invention is directed to a compound of Formula I ##STR00001## or a pharmaceutically acceptable salt thereof, wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4...
US-9,359,335 Triazole derivative, and light-emitting element, light-emitting device, electronic device and lighting device...
Objects are to provide the following: a substance that facilitates hole injection and has high triplet excitation energy; a light-emitting element having high...
US-9,359,334 Ligands for sensitizing dyes of dye-sensitized solar cells
The present invention provides new bi- and polypyridine ligands of ruthenium dyes. The invention also provides solar cells, in particular dye-sensitized solar...
US-9,359,333 Efficient process for the preparation of Lapatinib and salts thereof by means of new intermediates
The present invention refers to a new efficient process for the synthesis of the active pharmaceutical ingredient Lapatinib and salts thereof. In particular,...
US-9,359,332 Processes for the preparation of substituted quinazolines
The present disclosure provides compounds for modulating receptor kinase activity, particularly ephrin and EGFR, and methods of treating diseases mediated by...
US-9,359,330 Substituted piperidines as sodium channel blockers
The present disclosure provides substituted piperidines or pyrrolidines having Formula IA: ##STR00001## and the pharmaceutically acceptable salts and solvates...
US-9,359,329 Derivatives of 2-pyridin-2-yl-pyrazol-3(2H)-one, preparation and therapeutic use thereof
The invention relates to compounds corresponding to formula (I), in the form of the base or of an acid-addition salt: ##STR00001## in which n is equal to 0,...
US-9,359,328 2-[[[2-[(hydroxyacetyl)amino]-4-pyridinyl]methyl]thio]-N-[4-(trifluorometh- oxy)phenyl]-3-pyridinecarboxamide...
In the course of developing 2-[[[2-[(hydroxyacetyl) amino]-4-pyridinyl]methyl]thio]-N-[4-(trifluoromethoxy) phenyl]-3-pyridinecarboxamide(compound A), there are...
US-9,359,327 Process for the preparation of substituted pyrimidine derivatives
The present invention is directed to processes for the preparation of substituted pyrimidine derivatives, useful as intermediates in the synthesis of histamine...
US-9,359,326 Manufacturing process for pyrimidine derivatives
The invention relates to processes for manufacturing a compound of formula 5, ##STR00001## or a stereoisomer, tautomer or a salt thereof, wherein the...
US-9,359,325 Lipoyl compounds and methods for treating ischemic injury
The present invention relates, in various embodiments, to a compound represented by Structural Formula (I), pharmaceutically acceptable salts or prodrugs...
US-9,359,324 Process for preparing episulfide compounds
Provided is a method for producing an episulfide compound, the method including a step of thiating epoxy groups of (B) an epoxy compound by a reaction with (C)...
US-9,359,323 Compound
The present invention provides compounds of the formula Formula I or a salt thereof: and the uses of such compounds for the treatment of a disease or disorder...
US-9,359,322 C-linked glucuronide of N-(4-hydroxybenzyl) retinone, analogs thereof, and methods of using the same to inhibit...
Compounds of the formula: ##STR00001## are described, along with pharmaceutical compositions containing these compounds, and methods of using the compounds to...
US-9,359,321 Hydroxymethylfurfural derivative
The hydroxymethylfurfural derivative is represented by the general formula (A) (wherein, R is selected from the group consisting of the following formula (I),...
US-9,359,320 Acid-functionalized polyolefin materials and their use in acid-promoted chemical reactions
An acid-functionalized polyolefin material that can be used as an acid catalyst in a wide range of acid-promoted chemical reactions, wherein the ...
US-9,359,319 Hydrogenation of biomass-derived substrates
The .alpha.,.beta.-unsaturated ketone moiety of a substrate representative of non-food based biomass was hydrogenated to the corresponding saturated alcohol...
US-9,359,318 Process for the synthesis of 2,5-furandicarboxylic acid
Process for the synthesis of 2,5-furandicarboxylic acid through the oxidation of -hydroxymethylfurfural in a flow of oxygenor a compound containing oxygen,...
US-9,359,317 Small molecule inhibitors of HIV proteases
Described herein are compounds, compositions, and methods for treating HIV and related diseases.
US-9,359,316 Prodrugs of phenolic TRPV1 agonists
Described herein are compounds, pharmaceutical compositions and medicaments that include such compounds, and methods of using such compounds to modulate...
US-9,359,315 Substituted 2,3-dihydro-1H-inden-1-one retinoic acid-related orphan nuclear receptor antagonists for treating...
The present invention is directed to compounds, their synthesis, and their use as antagonists, inverse agonists, modulators and or inhibitors of the Retinoic...
US-9,359,314 Thiazine amide derivative and pharmaceutical composition and use thereof
The present invention relates to a thiazine amide derivative and a pharmaceutical use thereof, and particularly to a compound of formula I (in the formula,...
US-9,359,313 Use of metformin in combination with a glucokinase activator and compositions comprising metformin and a...
The present invention provides uses of a glucokinase activator in combination with metformin. Uses include treating type 2 diabetes, lowering blood glucose,...
US-9,359,312 Process for manufacturing benzoxazinones
The present invention relates to a process for manufacturing a benzoxazinone of formula (I), ##STR00001## by reacting a nitro compound of formula (II) with a...
US-9,359,311 Substituted aromatic oligomers
The present invention relates to novel chemical compounds formula (I) (C).sub.n--B-(A).sub.m-B--(C).sub.n (I) wherein m is 0 or 1, and n is independently 0, 1,...
US-9,359,310 Methanethione compounds having antiviral activity
A compound of formula (I) is useful as an antiviral agent, in particular for the treatment of influenza. A method for preparing the compound of formula (I) and...
US-9,359,309 Synthesis of syrbactin proteasome inhibitors
The disclosure relates generally to methods for the preparation of a family of natural compounds, the syrbactins and their analogs.
US-9,359,308 Pyrazine kinase inhibitors
Provided are pyrazine compounds of Formula (I) ##STR00001## for inhibiting of Syk kinase, intermediates used in making such compounds, methods for their...
US-9,359,306 Process for preparing pan-CDK inhibitors of the formula (I), and intermediates in the preparation
The invention relates to a novel process for the preparation of pan-CDK inhibitors of the formula (I), and intermediates of the preparation. ##STR00001##
US-9,359,305 Parasiticidal compositions comprising benzimidazole derivatives, methods and uses thereof
The invention relates to oral, topical or injectable compositions for combating liver fluke parasites in mammals, comprising at least one benzimidazole...
US-9,359,304 Process for the preparation of 3-haloalkylpyrazoles
The present invention provides a process for the preparation of a compound of formula (I) wherein R.sup.1 is C.sub.1-C.sub.4 haloalkyl; R.sup.2 is optionally...
US-9,359,303 Octahydrobenzoisoquinoline modulators of dopamine receptors and uses therefor
Octahydrobenzoisoquinoline modulators of dopamine receptors are described herein. Methods for using octahydrobenzoisoquinoline modulators of dopamine receptors...
US-9,359,302 Low hygroscopic aripiprazole drug substance and processes for the preparation thereof
The present invention provides low hygroscopic forms of aripiprazole and processes for the preparation thereof which will not convert to a hydrate or lose their...
US-9,359,301 Ethynyl derivatives
The present invention relates to ethynyl derivatives of formula I ##STR00001## wherein Y is N or CH R.sup.1 is fluoro or chloro or to a pharmaceutically...
US-9,359,300 Methyl/difluorophenyl-methoxy substituted pyridinone-pyridinyl compounds, methyl-pyridinyl-methoxy substituted...
The present disclosure provides methyl/difluorophenyl-methoxy substituted pyridinone-pyridinyl compounds, methyl-pyridinyl-methoxy substituted ...
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