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Patent # Description
US-9,428,504 7-hydroxy-spiropipiperidine indolinyl antagonists of P2Y.sub.1 receptor
The present invention provides compounds of Formula (I): as defined in the specification and compositions comprising any of such novel compounds. These...
US-9,428,503 Imidazo[4,5-c]quinolin-2-one compounds and their use in treating Cancer
The specification generally relates to compounds of Formula (I): ##STR00001## and pharmaceutically acceptable salts thereof, where Q, R.sup.1, R.sup.2,...
US-9,428,502 Heterocyclic modulators of lipid synthesis
Heterocyclic modulators of lipid synthesis are provided as well as pharmaceutically acceptable salts thereof; pharmaceutical compositions comprising such...
US-9,428,501 Bicyclic nitrogen-containing aromatic heterocyclic amide compound
Compounds of formula (I) and salts thereof: ##STR00001## wherein the variables are defined herein, are useful for the treatment of breast cancer.
US-9,428,500 Alpha-carbolines for the treatment of cancer
The present invention relates to inhibitors of the oncogenic protein kinase ALK of formula (I) as herein described and pharmaceutical compositions thereof, as...
US-9,428,499 Heterocyclyl compounds as MEK inhibitors
The present disclosure is related to heteroaryl compounds as MEK inhibitors. These compounds include heteroaryl compounds of formula I, their pharmaceutically...
US-9,428,498 Substituted imidazo[4,5-c]pyridine compounds and compositions thereof
The present invention relates to compounds which are inhibitors of SSAO activity. The invention also relates to pharmaceutical compositions comprising these...
US-9,428,497 Precursor compounds for the radiosynthesis of [.sup.18F] norchloro-fluorohomoepibatidine
The invention relates to a compound of formula Ia or Ib wherein R.sup.1 represents --CO.sub.2R.sup.3, --COR.sup.4 or --R.sup.5, wherein R.sup.3 represents...
US-9,428,496 Thiazolamine derivative and use thereof as anti-picornaviral infection medicament
Disclosed is as a substituted thiazolamine derivative represented by Formula I or a pharmaceutically acceptable salt thereof or a hydrate thereof (the...
US-9,428,495 Selectively substituted quinoline compounds
Embodiments of the disclosure relate to selectively substituted quinoline compounds that act as antagonists or inhibitors for Toll-like receptors 7 and/or 8,...
US-9,428,494 Therapeutic compounds
The invention provides novel compounds of formula I: that are opioid receptor ligands. The invention also provides pharmaceutical compositions comprising such...
US-9,428,493 Schweinfurthin analogues
The invention provides a compound of formula (I): wherein R.sup.1-R.sup.5 have any of the values defined in the specification. The compounds are useful for the...
US-9,428,492 Secondary alcohol substituted triazoles as PDE10 inhibitors
The present invention is directed to secondary alcohol substituted triazole compounds which are useful as therapeutic agents for the treatment of central...
US-9,428,491 Substituted azoles, antiviral active component, pharmaceutical composition, method for preparation and use thereof
The present invention relates to novel antiviral active 5-{4-[1H-imidazol-5-ylaryl(or hetaryl)]-buta-1,3-diynyl}-1H-imidazoles of the general formula 1 and...
US-9,428,490 Nuclear transport modulators and uses thereof
The invention generally relates to nuclear transport modulators, e.g CRM1 inhibitors, and more particularly to a compound represented by formula (I): or a...
US-9,428,489 Benzimidazole-carboxamide compounds as 5-HT.sub.4 receptor agonists
The invention relates to benzimidazole-carboxamide 5-HT.sub.4 receptor agonist compounds of formula (I) ##STR00001## wherein R.sup.1 and X are as defined in...
US-9,428,488 Method for producing 4-[5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl]pyridine-2-carbonitrile, and intermediate...
To provide an industrially useful method for producing pharmaceutically useful 4-[5-(pyridin-4-yl)-1H-1,2,4-triazol-3-yl]pyridine-2-carbonitrile, and an...
US-9,428,487 Heteroaromatic amides and thioamides as pesticides
The present application relates to novel amides and thioamides, to processes for preparation thereof and to use thereof for controlling animal pests, in...
US-9,428,486 Efficient process for the preparation of Esomeprazole (S)-Binol complex
Object of the present invention is an improved process for the preparation of Esomeprazole (S)-BINOL complex which is a key intermediate for the synthesis of...
US-9,428,485 Salt, photoresist composition and method for producing photoresist pattern
A salt represented by formula (I): ##STR00001## wherein Q.sup.1 and Q.sup.2 each independently represent a fluorine atom or a C1-C6 perfluoroalkyl group,...
US-9,428,484 Method for the production of cyclic diesters, in particular dilactide
The present invention relates to a method for the production of cyclic carboxylic acid esters, in particular intramolecular lactones, such as e.g. dilactide,...
US-9,428,483 Prodrug of fluorine-containing amino acid
Provided are a fluorine-containing amino acid prodrug represented by general formula (I) that makes a fluorine-containing amino acid which is a group 2...
US-9,428,482 Process for synthesis of polyphenols
The present invention provides synthetic processes for preparing racemic and/or optically pure epicatechin, epigallocatechin and related polyphenols as such or...
US-9,428,481 Process for the preparation of 2 substituted tetrahydropyranols
The present invention relates to a process for the preparation of 2-substituted 4-hydroxy-4-methyltetrahydropyrans by reacting 3-methylbut-3-en-1-ol (isoprenol)...
US-9,428,480 Oxidation process to produce a crude and/or purified carboxylic acid product
Disclosed is an oxidation process to produce a crude carboxylic acid product carboxylic acid product. The process comprises oxidizing a feed stream comprising...
US-9,428,479 Conversion of biomass
Biomass feedstocks (e.g., plant biomass, animal biomass, and municipal waste biomass) are processed to produce useful products, such as fuels. For example,...
US-9,428,478 Piperazine derivatives, compositions, and uses related thereto
The disclosure relates to piperazine derivatives, compositions, and methods related thereto. In certain embodiments, the disclosure relates to inhibitors of...
US-9,428,477 Trans-2-decenoic acid derivative and drug containing same
The present invention relates to a novel trans-2-decenoic acid derivative or a pharmaceutically acceptable salt thereof, and a pharmaceutical agent containing...
US-9,428,476 S-imino-S-oxo-iminothiadiazine compounds as BACE inhibitors, compositions, and their use
In its many embodiments, the present invention provides provides certain S-imino-S-oxo iminothiadiazine compounds, including compounds Formula (I): or a...
US-9,428,475 Iminothiadiazine dioxide compounds as BACE inhibitors, compositions, and their use
In its many embodiments, the present invention provides certain iminothiadiazine dioxide compounds, including compounds Formula (I): (I) and include...
US-9,428,474 Antibacterial compounds
The present invention relates to the following compounds for use in the treatment of a bacterial infection ##STR00001## wherein the integers are as defined in...
US-9,428,473 Methods and intermediates for preparing pharmaceutical agents
The invention provides methods and intermediates that are useful for preparing a compound of formula I: ##STR00001## and salts thereof.
US-9,428,472 Methods of treating bacterial infections with 1,2-benzisothiazolinone and isoindolinone derivatives
Methods of treating, preventing and ameliorating bacterial infections with 1,2-benzisothiazolinone and isoindolinone derivatives are disclosed. Pharmaceutical...
US-9,428,471 Cyclic carbamate compounds useful in energy-curable compositions
Cyclic carbamate functional compounds, which are the reaction product of a cyclic carbamate having an acrylate functional group, such as ...
US-9,428,470 Heterocyclic compound
A fused heterocyclic compound having an enteropeptidase inhibitory action and use of the compound as a medicament for treatment or prophylaxis of obesity,...
US-9,428,469 Antiviral compounds
The present invention discloses compounds of Formula (I): wherein the variables in Formula I are defined as described herein. Also disclosed are pharmaceutical...
US-9,428,468 Process for the preparation of erlotinib
A process for the preparation of Erlotinib is disclosed in which the compound of formula (II) ##STR00001## Is reacted with the compound of formula (III) in...
US-9,428,467 Selective calcium channel antagonists
The present invention relates to compositions and methods for the treatment and/or prevention of neurodegenerative disorders, e.g., Parkinson's disease (PD). In...
US-9,428,466 Methods for reducing uric acid levels using barbiturate derivatives
Methods for reducing uric acid levels in blood or serum of a subject employing metabolites of merbarone as active agents. Methods for treating or preventing...
US-9,428,465 Acid ceramidase inhibitors and their use as medicaments
The present invention concerns, in a first aspect, compounds of Formula I as defined herein, pharmaceutically acceptable salts thereof and pharmaceutical...
US-9,428,464 Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof
Certain chemical entities are provided herein. Also provided are pharmaceutical compositions comprising at least one chemical entity and one or more...
US-9,428,463 N.sup..alpha., N.sup..alpha., N.sup..alpha.-trialkyl histidine derivatives useful for the preparation of...
Provided herein are N.sup..alpha.,N.sup..alpha.,N.sup..alpha.-trialkyl histidine derivative compounds and methods of their preparation. Also provided are...
US-9,428,462 4-[-2-[[5-methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine hydrochloride amorphous solid forms
The present invention relates to solid forms having a low degree of crystallinity or substantially amorphous of the hydrochloride salt of ...
US-9,428,461 Process for the preparation of a benzazepine derivative
Provided is an industrially scalable process for the preparation of a benzazepine derivative, namely, 7-chloro-5-hydroxy-1-[2-methyl-4-(2-methyl benzoyl amino) ...
US-9,428,460 N-[4-(quinolin-4-yloxy)cyclohexyl(methyl)](hetero)arylcarboxamides as androgen receptor antagonists, production...
The invention relates to N-[4-(quinolin-4-yloxy)cyclohexyl(methyl)](hetero)arylcarboxamides, intermediates and methods for their production, use thereof for...
US-9,428,459 Difluoromethyl-nicotinic- tetrahydronaphtyl carboxamides
The present invention relates to novel difluoromethyl-nicotinic indanyl carboxamide compounds, to processes for preparing the carboxamide compounds, to...
US-9,428,458 Substituted pyridoxine-lactam carboxylate-salts
The present invention provides salt adducts comprising at least one positively charged moiety being a pyridoxine or a derivative thereof and at least one...
US-9,428,457 Neprilysin inhibitors
In one aspect, the invention relates to compounds having the formula: ##STR00001## where R.sup.1-R.sup.5 and X are as defined in the specification, or a...
US-9,428,456 1-[m-carboxamido(hetero)aryl-methyl]-heterocyclyl-carboxamide derivatives
The present invention relates to 1-[m-carboxamido(hetero)aryl-methyl]-heterocycyl-carboxamide compounds of formula (I) ##STR00001## wherein X, Ar.sup.1,...
US-9,428,455 Process for annealing amorphous atorvastatin
Processes for annealing amorphous atorvastatin is described. Pharmaceutical compositions and formulations containing annealed amorphous atorvastatin are also...
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