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Patent # Description
US-9,487,526 Quinoxaline derivatives as GPR6 modulators
The present invention provides compounds of Formula (I): ##STR00001## that are GPR6 modulators and are therefore useful for the treatment of diseases treatable...
US-9,487,525 Crystalline forms of (s)-4-amino-n-(1-(4-chlorophenyl)-3-hydroxypropyl)-1-(7h-pyrrolo[2,3-d]py- ...
The present invention discloses certain new solid state forms of (S)-4-amino-N-(1-(4-chlorophenyl)-3-hydroxypropyl)-1-(7H-pyrrolo[2,3-d]py- ...
US-9,487,524 Phenyl-urea and phenyl-carbamate derivatives as inhibitors of protein aggregation
The present invention relates to certain phenyl-urea and phenyl-carbamate derivatives comprising a bicyclic heteroaryl group, pharmaceutical compositions...
US-9,487,523 Process for making CGRP receptor antagonists
The invention encompasses a novel process for making piperidinone carboxamide indane and azainane derivatives, which are CGRP receptor antagonists useful for...
US-9,487,522 SSH-2 (slingshot-2) inhibitors and methods for making and using them
In alternative embodiments, the invention provides compositions that inhibit the polypeptide SSH-2, or SlingSHot-2, a phosphatase enzyme that regulates actin...
US-9,487,521 Processes and intermediates for making a JAK inhibitor
This invention relates to processes and intermediates for making {1-{1-[3-fluoro-2-(trifluoromethyl)isonicotinoyl]piperidin-4-yl}-3-[4-(7H- ...
US-9,487,520 Coelenterazine derivatives and methods of using same
The invention provides coelenterazine derivatives which are substrates for a non-luminescent enzyme and a pro-substrate for a luminescent enzyme. The invention...
US-9,487,519 5,6-Dialkyl-7-aminotriazolopyrimidines, their preparation and their use for controlling harmful fungi, and...
5,6-Dialkyl-7-aminotriazolopyrimidines of the formula I ##STR00001## in which the substituents are as defined below: R.sup.1 is alkyl or alkoxyalkyl, where...
US-9,487,518 HIV inhibiting bicyclic pyrimidine derivatives
HIV replication inhibitors of formula ##STR00001## wherein -a.sup.1=a.sup.2-a.sup.3=a.sup.4- is --CH.dbd.CH--CH.dbd.CH--, --N.dbd.CH--CH.dbd.CH--,...
US-9,487,517 Spiroimidazolone derivative
The present invention relates to a compound represented by the following formula (1): ##STR00001## wherein W, X, Y, R.sub.1, R.sub.2, R.sub.33, R.sub.34, m...
US-9,487,516 Antibacterial oxadiazolone derivatives
The invention relates to antibacterial compounds of formula I ##STR00001## wherein U represents CH or N; V represents CH or N, provided that at least one of U...
US-9,487,515 Compounds modulating c-fms and/or c-kit activity and uses therefor
Compounds active on the receptor protein tyrosine kinases c-kit and/or c-fms are provided herewith. Also provided herewith are compositions useful for treatment...
US-9,487,514 Neprilysin inhibitors
In one aspect, the invention relates to compounds having the formula: ##STR00001## where R.sup.1, R.sup.2a, R.sup.2b, R.sup.3--R.sup.6, a, b, Z, and X are as...
US-9,487,513 Substituted pyrazolo[1,5-A]pyridines, their preparation and use as medicaments
The present invention relates to new substituted pyrazolo[1,5-a]pyridine having a great affinity for sigma receptors, especially sigma-1 receptor, as well as to...
US-9,487,512 (Hetero)aryl cyclopropylamine compounds as LSD1 inhibitors
The invention relates to (hetero)aryl cyclopropylamine compounds, including particularly the compounds of formula I as described and defined herein, and their...
US-9,487,511 Cyclopropanamine compound and use thereof
The present invention provides a compound having a lysine-specific demethylase-1 inhibitory action, and useful as a medicament such as a prophylactic or...
US-9,487,510 Substituted heterocyclic acetamides as kappa opioid receptor (KOR) agonists
The present invention relates to a series of substituted compounds having the general formula (I), including their stereoisomers and/or their pharmaceutically...
US-9,487,509 Heterocyclic compound
The present invention relates to ##STR00001## wherein each symbol is as defined in the specification. The compound of the present invention has a superior...
US-9,487,508 SGC stimulators
The present patent application discloses at least the compounds according to Formula I or Formula Ib shown below, or pharmaceutically acceptable salts thereof, ...
US-9,487,507 TRPV4 antagonists
The present invention relates to spirocarbamate analogs, pharmaceutical compositions containing them and their use as TRPV4 antagonists.
US-9,487,506 Mineralocorticoid receptor antagonists
Compounds of the Formula (I) as well as pharmaceutically acceptable salts thereof, that may be useful for treating aldosterone-mediated diseases are disclosed....
US-9,487,505 Heteroaryl-substituted 1,3-dihydroindol-2-one derivatives and medicaments containing them
The present invention relates to novel 1,3-dihydroindol-2-one (oxindole) derivatives of the formula (I) ##STR00001## in which A, R.sup.3, R.sup.4, R.sup.5,...
US-9,487,504 Imidazolyl analogs as syk inhibitors
The present invention provides novel imidazole analogs of Formula I which are potent inhibitors of spleen tyrosine kinase, and are useful in the treatment and...
US-9,487,503 Stilbene optical brighteners
The present invention discloses compounds of 4,4'-diaminostilbene-2,2'-disulphonic acid which are useful as optical brighteners to bleach fibers, cellulose and...
US-9,487,502 Chemical compounds
The invention relates to pyrrolone compounds of the formula (I) wherein X, R.sup.1, R.sup.2, R.sup.3, R.sup.a, R.sup.c and R.sup.d are as defined in the...
US-9,487,501 Pyrazole carboxamide compounds and uses thereof
The present invention relates to compounds of formula ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, and Z are as descried in the claims, or to a...
US-9,487,500 Compounds and compositions thereof
Novel compounds and their synthesis are described. Methods for using these compounds in the prevention or treatment of cancer, a bacterial infection or a viral...
US-9,487,499 Methods of making fused ring compounds
The present invention relates to methods of making fused ring compounds, such as indeno-fused naphthols, and fused ring indenopyran compounds, such as...
US-9,487,498 N-hydroxylsulfonamide derivatives as new physiologically useful nitroxyl donors
The invention relates to N-hydroxysulfonamide derivatives that donate nitroxyl (HNO) under physiological conditions and are useful in treating and/or preventing...
US-9,487,497 Synthetic process for preparing 2-((2-ethoxy-2-oxoethyl)(methyl)amino)-2-oxoethyl ...
Disclosed herein are processes for forming 2-((2-ethoxy-2-oxoethyl)(methyl)amino)-2-oxoethyl 5-tetradecyloxy)furan-2-carboxylate: ##STR00001##
US-9,487,496 Process for the preparation of cabazitaxel and its intermediates
The present invention relates to a novel process for preparation of cabazitaxel (I) starting from 10-Deacetyl baccatin or derivative that involves methylation...
US-9,487,495 Carbamate compounds and of making and using same
This disclosure provides compounds having the structure: ##STR00001## wherein L.sup.3, R.sup.7, R.sup.d and p are defined herein, which are modulators of MAGL...
US-9,487,494 Cyclic hydrocarbon compounds for the treatment of diseases
The invention relates to novel cyclic hydrocarbon compounds and derivatives thereof, processes for the preparation thereof, to said compounds for use as a...
US-9,487,493 Use of a PPAR-delta agonist for treating muscle atrophy
The present invention provides methods for treating muscle atrophy by administering a PPAR.delta. agonist.
US-9,487,492 Dibenzothiazepine derivatives and their use in the treatment of CNS disorders
A compound of formula I: ##STR00001## or a pharmaceutically or veterinarily acceptable salt thereof, or a pharmaceutically or veterinarily acceptable solvate...
US-9,487,491 Diamino heterocyclic carboxamide compound
Provided is a compound useful as an inhibitor against the kinase activity of EML4-ALK fusion protein. As a result of intensive and extensive studies on...
US-9,487,490 3-cyclohexenyl and cyclohexyl substituted indole and indazole compounds as RORgammaT inhibitors and uses thereof
The present invention relates to compounds according to Formula I and pharmaceutically acceptable salts or solvates thereof. Such compounds can be used in the...
US-9,487,489 Halogen-substituted pyrazole derivatives as pest-control agents
The invention relates inter alia to halogen-substituted compounds of the general formula (I) ##STR00001## in which the radicals A.sub.1-A.sub.4, T, n, W, Q,...
US-9,487,488 Sulfonamide compound
The present invention provides novel sulfonamide compounds having TRPM8 antagonistic activity which are useful as medicaments. Specifically, the present...
US-9,487,487 Process for preparation of montelukast sodium
Disclosed is a process for the preparation of montelukast sodium. The process comprises a) reacting ...
US-9,487,486 Derivatives of nicotinic acid N-oxide, their preparation and their use as inhibitors of enzyme...
A derivative of nicotinic acid N-oxide is described having formula (I): that acts as inhibitor of enzyme 3-hydroxyanthranilate-3,4-dioxygenase (3HAO), and is...
US-9,487,485 Method for producing sulfonyl chloride compound
An object of the present invention is to provide a production method of an intermediate used in the production method of a sulfonylpyrrole compound useful as a...
US-9,487,484 Stilbazolium derivative and nonlinear optical material using the same
Provided is a stilbazolium derivative represented by the general formula (I): ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, and R.sup.4 independently...
US-9,487,483 Complement pathway modulators and uses thereof
The present invention provides a compound of formula (I): a method for manufacturing the compounds of the invention, and its therapeutic uses. The present...
US-9,487,482 3,4,5-trimethoxystyrylarylaminopropenones as potential anticancer agents
The present invention relate to compounds of general formula A. The invention also provides the synthesis of 3,4,5-trimethoxystyrylarylaminopropenones useful as...
US-9,487,481 Bicyclic compounds
Disclosed are compounds of Formula (I) ##STR00001## and/or a salt thereof; wherein R is --OH or --OP(O)(OH).sub.2. Also disclosed are methods of using such...
US-9,487,480 Zwitterionic reagents
Zwitterion-containing compounds for the modification of hydrophobic molecules to improve their solubility and/or to lower their non-specific binding as...
US-9,487,479 Small molecule inhibitors of N-terminus activation of the androgen receptor
Compounds having a structure of Formula (A) are provided. Uses of such compounds for treatment of various indications, including prostate cancer as well as...
US-9,487,478 Difluorolactam compounds as EP4 receptor-selective agonists for use in the treatment of EP4-mediated diseases...
Disclosed herein are compounds of formula (I) ##STR00001## and therapeutic methods of treatment with compounds of formula (I), wherein L.sup.1, L.sup.2,...
US-9,487,477 Crystalline phase of (3S,3S') 4,4'-disulfanediylbis(3-aminobutane 1-sulfonic acid) with L-lysine
The present invention relates to a new crystalline phase of (3S,3S') 4,4'-disulfanediylbis(3-aminobutane 1-sulfonic acid) (ABSD) with L-lysine and its use,...
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