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Patent # Description
US-9,499,566 Oxidation process for preparing 3-formyl-cephem derivatives
The present invention relates to an improved process for oxidizing 3-hydroxy-methyl-cephem derivatives to the corresponding 3-formyl-cephem derivatives. In...
US-9,499,565 Cocrystal of piperacillin sodium and sulbactam sodium and preparation method thereof, as well as pharmaceutical...
Provided in the present invention are a cocrystal of piperacillin sodium and sulbactam sodium and preparation method thereof, as well as pharmaceutical...
US-9,499,564 CDK inhibitors
Compounds of formulae I, II or III, and pharmaceutically acceptable salts thereof, are useful as CDK inhibitors.
US-9,499,563 Thieno [2, 3-B] pyridine derivatives as viral replication inhibitors
The present invention relates to a series of compounds having antiviral activity, more specifically HIV (Human Immunodeficiency Virus) replication inhibiting...
US-9,499,562 Substituted thiophene- and furan-fused azolopyrimidine-5-(6H)-one compounds
Described herein are compounds and chemical entities of Formula (I), methods of their synthesis, compositions comprising them, and their use in treating...
US-9,499,561 Fused pyrimidine compound, and preparation method, intermediate, composition, and uses thereof
Disclosed are a fused pyrimidine compound as represented by formula I, pharmaceutically acceptable salt, hydrate and solvate thereof, an optical isomer or a...
US-9,499,560 N-containing heterocyclic compounds
The present invention relates to N-containing heterocyclic compounds that are inhibitors of protein kinases including JAK kinases. In particular, the compounds...
US-9,499,559 Method for preparing long-chain alkyl cyclic acetals made from sugars
Long-chain alkyl cyclic acetals made from sugars are obtainable by a method that comprises the steps consisting of: dehydrating a hexitol in a...
US-9,499,558 Compounds and methods for treating HIV
Inhibitors of HIV-1 protease and compositions containing them are described. Use of the inhibitors and compositions containing them to treat HIV, AIDS, and...
US-9,499,557 Transition metal-catalyzed processes for the preparation of N-allyl compounds and use thereof
The present disclosure provides processes for the N-dealkylation of tertiary amines and the use of transition metal catalysts to prepare tertiary N-allyl amine...
US-9,499,556 Convenient preparation of N-substituted morphinan-6-ols from morphinan-6-ones
Described herein are methods of preparing 6-hydroxy N-alkyl morphinan-6-ols from morphinan-6-ones, as illustrated below: ##STR00001## wherein the variables...
US-9,499,555 Porous crystalline frameworks, process for the preparation therof and their mechanical delamination to covalent...
The invention disclosed herein provides, Porous Crystalline Frameworks (PCFs) also known as Covalent Organic Frameworks (COFs) that exhibit stability towards...
US-9,499,554 Anti-influenza compositions and methods
Disclosed are novel compounds comprising an imino-ribose derivative covalently linked to a carbocycle or heterocycle. Pharmaceutical compositions comprising the...
US-9,499,553 Dihydropyridazine-3,5-dione derivative and pharmaceuticals containing the same
The present invention provides a dihydropyridazine-3,5-dione derivative or a salt thereof, or a solvate of the compound or the salt, a pharmaceutical drug, a...
US-9,499,552 Pyrazolo[1,5-A]pyrimidine derivative and use of anti-tumor thereof
The present invention relates to a pyrazolo[1,5-a]pyrimidine derivative of general formula 1 and a pharmaceutically acceptable salt thereof. The present...
US-9,499,551 Substituted pyrrolo[2,3-b]pyridines for treating cancer or inflammatory diseases
Disclosed herein are substituted pyrrolopyridine and pyrrolopyrazine compounds and compositions useful in the treatment of TAK mediated diseases, such as...
US-9,499,550 Hepatitis C virus inhibitors
Hepatitis C virus inhibitors having the general formula (I) are disclosed. Compositions comprising the compounds and methods for using the compounds to inhibit...
US-9,499,549 Pyrrolo[3,2-]pyrimidine derivatives for the treatment of viral infections and other diseases
This invention concerns pyrrolo[3,2-d]pyrimidine derivatives, processes for their preparation, pharmaceutical compositions, and their use in treatment and/or...
US-9,499,548 Inhibitors of bruton's tyrosine kinase
This application discloses compounds according to generic Formula I: wherein all variables are defined as described herein, which inhibit Btk. The compounds...
US-9,499,547 Amino-substituted imidazopyridazines
The present invention relates to amino-substituted imidazopyridazine compounds of general formula (I): in which A, R1, R3 and n are as defined in the claims, to...
US-9,499,546 Process for the preparation of chiral 8-(3-aminopiperidin-1-yl)-xanthines
The invention relates to an improved process for preparing enantiomerically pure 8-(3-aminopiperidin-1-yl)-xanthines.
US-9,499,545 Piperidinone carboxamide azaindane CGRP receptor antagonists
The present invention is directed to piperidinone carboxamide azaindane derivatives which are antagonists of CGRP receptors and useful in the treatment or...
US-9,499,544 Nitrogen containing heterocyclic compounds
Compounds of Formula (I), their preparation and use in preventing or treating bacterial infections are disclosed. ##STR00001##
US-9,499,543 Polymorph forms
The present invention relates to novel crystal forms of 2-amino-N-[2-(3a-(R)-benzyl-2-methyl-3-oxo-2,3,3a,4,6,7-hexahydro-pyrazol- ...
US-9,499,542 Arylpyrrolopyridine derived compounds as LRRK2 inhibitors
The present invention is directed to arylpyrrolopyridine derivatives of formula (A) (A). The compounds are considered useful for the treatment of diseases...
US-9,499,541 Piperidinone carboxamide indane CGRP receptor antagonists
The present invention is directed to piperidinone carboxamide indane derivatives which are antagonists of CGRP receptors and useful in the treatment or...
US-9,499,540 Purified pyrroloquinolinyl-pyrrolidine-2,5-dione compositions and methods for preparing and using same
The present invention relates to a (.+-.)-trans-3-(5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinolin-1-yl)-4-(1H-indo- l-3-yl)pyrrolidine-2,5-dione dichloromethane.
US-9,499,539 Cyclic sulfonamide containing derivatives as inhibitors of hedgehog signaling pathway
The invention relates generally to the creation and use of cyclic sulfonamide containing derivatives to inhibit the hedgehog signaling pathway and to the use of...
US-9,499,538 Estrogen receptor modulators and uses thereof
Described herein are compounds that are estrogen receptor modulators. Also described are pharmaceutical compositions and medicaments that include the compounds...
US-9,499,537 Antiviral pyrrolopyridine derivatives and method for preparing the same
The present invention relates to a pyrrolopyridine derivative represented by the Chemical Formula I, and a racemate or a stereoisomer thereof, or a ...
US-9,499,536 Tetrahydro-pyrido-pyrimidine derivatives
The invention relates to substituted tetrahydro-pyrido-pyrimidine derivatives of the formula (I), ##STR00001## wherein Y, R.sup.1, R.sup.2 and m are as...
US-9,499,535 Kinase inhibitors
The present invention relates to novel compounds of formula (I) ##STR00001## that are capable of inhibiting one or more kinases, especially SYK (Spleen...
US-9,499,534 Thiazole-substituted aminopyrimidines as spleen tyrosine kinase inhibitors
The invention provides certain thiazole-substituted aminopyrimidine compounds of the Formula (I) (I), or pharmaceutically acceptable salts thereof, wherein R1,...
US-9,499,533 Aromatic 5-membered heterocyclic derivative having TRPV4-Inhibiting activity
The present invention is related to a compound represented by formula (I) ##STR00001## wherein R.sup.1 is a hydrogen atom, substituted or unsubstituted alkyl,...
US-9,499,532 Therapeutic compounds and compositions
The present invention provides compounds and compositions that inhibit Factor XIa or kallikrein and methods of using these compounds and composition.
US-9,499,531 Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine,...
The compounds of the present invention are represented by the chemical structure found in Formula (I): ##STR00001## wherein: the carbon atom designated * is...
US-9,499,530 Quinazoline derivative, composition having the derivative, and use of the derivative in preparing medicament
A class of quinazoline derivatives or pharmaceutically acceptable salts or solvates thereof with novel structures is provided; meanwhile, a pharmaceutical...
US-9,499,529 Therapeutic uses of curcumin analogs for treatment of prostate cancer
This invention relates generally to methods of treating aggressive cancers, such as hormone-refractory metastatic prostate cancer, by exposing the aggressive...
US-9,499,528 Class of near infrared molecular probes for biological applications
Methods for preparing 2,5-Bis(benzoxazol-2'-yl)benzene-1,4-diol derivatives (Zinhbo derivatives) are provided. Zinhbo derivatives are used to detect zinc ions...
US-9,499,527 Compositions and methods for the treatment of familial amyloid polyneuropathy
The invention relates to the compounds of formula I or its pharmaceutical acceptable salts, as well as polymorphs, solvates, enantiomers, stereoisomers and...
US-9,499,526 Compositions and methods for the treatment of neurologic diseases
The invention relates to the compounds of formula I or its pharmaceutical acceptable salts, as well as polymorphs, solvates, enantiomers, stereoisomers and...
US-9,499,525 Dihydrate of benzothiophene compound or of a salt thereof, and process for producing the same
An object of the present invention is to provide a compound that can be used as a more superior therapeutic agent for central nervous system diseases. The...
US-9,499,524 Insecticidal compounds
The present invention relates to novel triazole derivatives of formula (I) having insecticidal activity, to processes and intermediates for preparing them, to...
US-9,499,523 Phosphatidylinositol 3-kinase inhibitors
The present application provides the compounds of formula (J), ##STR00001## or pharmaceutically acceptable salts, isomers, tautomer, or a mixture thereof,...
US-9,499,522 Compositions useful for treating disorders related to kit
Compounds and compositions useful for treating disorders related to Kit are described herein.
US-9,499,521 Inhibitors of cellular necrosis and related methods
A compound having the following structure (I): ##STR00001## or a pharmaceutically acceptable salt, prodrug, stereoisomer or tautomer thereof, is provided....
US-9,499,520 Process for the preparation of voriconazole and analogues thereof
The present invention provides a process for preparing a compound of formula: (Formula XI and XII) (XI) (XII) wherein X, Y, Z, A, B and E are as defined herein,...
US-9,499,519 Fused pyrimidine compounds and use thereof
Fused pyrimidine compounds as kinase inhibitors, such as multi-kinase inhibitors, are provided. Fused pyrimidine compounds as IGF-IR inhibitors are provided....
US-9,499,518 Bis-quaternary ammonium salts as pain modulating agents
Provided are methods for using bis-quaternary ammonium compounds to treat inflammatory pain, neuropathic pain and nociceptive pain.
US-9,499,517 Substituted prolines / piperidines as orexin receptor antagonists
The present invention is directed to compounds that modulate the bioactivity of an orexin receptor such as OX.sub.1 or OX.sub.2, or both; to pharmaceutical...
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