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Patent # Description
US-9,505,765 4-alkoxy/aralkoxy-5-substituted-pyrrolopyrimidine compounds as TAK1 inhibitors in disease treatment
4-alkoxy/aralkoxy-5-substituted-pyrrolopyrimidine compounds, pharmaceutically acceptable salts, solvates and pharmaceutical compositions of compounds embraced...
US-9,505,764 Treatment of cancer with dihydropyrazino-pyrazines
Provided herein are methods for treating or preventing chronic lymphocytic leukemia, comprising administering an effective amount of a Dihydropyrazino-Pyrazine...
US-9,505,763 Cancer treatment using BMP inhibitor
Methods for regulating cancer cell growth and survival, inhibiting cancer cell growth, promoting cancer cell death, and/or treating a cancer make use of...
US-9,505,762 Purine derivatives as CB2 receptor agonists
The invention relates to a compound of formula (I) ##STR00001## wherein A and R.sup.1 to R.sup.4 are defined as in the description and in the claims. The...
US-9,505,761 Bicyclic compounds and their use as antibacterial agents and beta-lactamase inhibitors
New bicyclic compounds, their preparation, and their use as antibacterial agents, either alone or in combination with an antibiotic for the treatment of...
US-9,505,760 Pyridopyrimidine based derivatives as potential phosphodiesterase 3 (PDE3) inhibitors and a process for the...
The present invention provides compounds of formula 1 as potential phosphodiesterase3 (PDE3) inhibitory agents and a process for the preparation thereof. The...
US-9,505,759 Pd-catalyzed coupling of pyrazole amides
A novel process for the preparation of imidazo[1,2-a]pyridine compounds of the formula ##STR00001## wherein R.sup.1 is C.sub.1-4-alkoxy or NR.sup.4R.sup.5...
US-9,505,758 Substituted 1,5-naphthyridines as endonuclease inhibitors
The present invention relates to a compound having the general formula (V), optionally in the form of a pharmaceutically acceptable salt, solvate, polymorph,...
US-9,505,757 Pharmaceutical composition comprising bicyclic pyridinol derivatives for preventing or treating diseases caused...
Disclosed is a pharmaceutical composition including a bicyclic pyridinol derivative as an active ingredient for preventing or treating diseases caused by...
US-9,505,756 Compounds useful for treating disorders related to TRPA1
Compounds and compositions for treating disorders related to TRPA1 are described herein.
US-9,505,755 Tetrahydropyrido-pyridine and tetrahydropyrido-pyrimidine compounds and use thereof as C5A receptor modulators
The present invention provides a compound of formula I: ##STR00001## a method for manufacturing the compounds of the invention, and its therapeutic uses. The...
US-9,505,754 Compound useful for the treatment of degenerative and inflammatory diseases
A compound is disclosed that has a formula represented by the following: ##STR00001## This compound may be prepared as a pharmaceutical composition, and may be...
US-9,505,753 Inhibitors of D-amino acid oxidase
D-amino acid oxidase (DAAO) inhibitors and methods of their use, either alone or in combination with D-serine or D-alanine, to facilitate allosteric activation...
US-9,505,752 Piperidine amide derivatives as HIV attachment inhibitors
Compounds of Formula I, including pharmaceutically acceptable salts thereof: formula (I): wherein A is selected from the group consisting of: formula (II) and...
US-9,505,751 Substituted [1,2,4]triazolo[1,5-a]pyrazines as phosphodiesterase inhibitors
Provided herein are substituted triazolopyrazine phosphodiesterase inhibitors, and pharmaceutical compositions thereof, useful for the treatment of, for...
US-9,505,750 5-aminocyclylmethyl-oxazolidin-2-one derivatives
The invention relates to antibacterial compounds of formula I ##STR00001## wherein one or two of U, V, W, and X represent N, the rest represent CH or, in the...
US-9,505,749 Quinazolinone compounds and derivatives thereof
Compounds of Formula I are useful inhibitors of tankyrase. Compounds of Formula I have the following structure: where the definitions of the variables are...
US-9,505,748 Amide-substituted heterocyclic compounds useful as modulators of IL-12, IL-23 and/or IFN.alpha. responses
Compounds having the following formula I: or a stereoisomer or pharmaceutically-acceptable salt thereof, where R.sup.1, R.sup.2, R.sup.3, R.sup.4, and R.sup.5...
US-9,505,747 Processes for preparing tubulysin derivatives and conjugates thereof
The invention described herein pertains to processes for preparing tubulysin derivatives, conjugates of tubulysins, and intermediates therefore. In one...
US-9,505,746 Pyrazol-4-yl-heterocyclyl-carboxamide compounds and methods of use
Pyrazol-4-yl-heterocyclyl-carboxamide compounds of Formula I, including stereoisomers, geometric isomers, tautomers, and pharmaceutically acceptable salts...
US-9,505,745 Enhancer of zeste homolog 2 inhibitors
This invention relates to novel compounds according to Formula (I) which are inhibitors of Enhancer of Zeste Homolog 2 (EZH2), to pharmaceutical compositions...
US-9,505,744 Solid state forms of vilazodone and vilazodone hydrochloride
The present invention provides solid state forms of Vilazodone and Vilazodone hydrochloride, processes for preparing these solid state forms, and pharmaceutical...
US-9,505,743 Matrix metalloproteinase inhibitors and methods for the treatment of pain and other diseases
The present invention relates generally to bis-amide containing MMP inhibiting compounds, and more particularly to selectively deuterated bis-amide MMP-13...
US-9,505,742 3,4-dihydro-2H-isoquinoline-1-one and 2,3-dihydro-isoindol-1-one compounds
The invention provides novel compounds having the general formula (I) ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, R.sup.7,...
US-9,505,741 Prolylhydroxylase inhibitors and methods of use
Compounds for inhibiting hypoxia inducible factor (HIF) prolyl-4-hydroxylases (PHDs) having the general formula (1). Methods of using these and related...
US-9,505,740 Cyclic amine derivative and pharmaceutical use thereof
A compound exerts a strong analgesic effect against pain, in particular, neuropathic pain and/or fibromyalgia syndrome. The cyclic amine derivative is...
US-9,505,739 Spiropyrrolidine beta-secretase inhibitors for the treatment of alzheimer's disease
The present invention is directed to spiropyrrolidine compounds of formula (I) which are inhibitors of the beta-secretase enzyme and that are useful in the...
US-9,505,738 Functional food additives
Novel compounds, and in particular to diacylglycerol (1, 3-DAG) and alpha-lipoic acid (LA) and/or dihydro-alpha-lipoic acid (DHLA) derivatives. In particular...
US-9,505,737 Treprostinil derivative compounds and methods of using same
Compounds represented by formulae I, II, III, and IV including pro-drugs for treprostinil and prostacyclin analogs. Uses include treatment of pulmonary...
US-9,505,736 Histone deacetylase inhibitors and compositions and methods of use thereof
Provided are certain histone deacetylase (HDAC) inhibitors of Formula I, compositions thereof, and methods of their use. ##STR00001##
US-9,505,735 Compounds for treating infectious diseases
The present invention provides compounds of Formula I, pharmaceutically acceptable salts thereof, and pharmaceutical compositions thereof. Compounds of the...
US-9,505,734 Phenyl C-glucoside derivative containing deoxyglucose structure, preparation method and use thereof
The present invention provides a phenyl C-glucoside derivative containing a deoxyglucose structure as represented by formula I, preparation method thereof, a...
US-9,505,733 Single step enantioselective process for the preparation of 3-substituted chiral phthalides
The present invention discloses single step, highly enantioselective catalytic oxidative cyclization process for the synthesis of 3-substituted chiral...
US-9,505,732 Auto magnetic metal salen complex compound
A drug using the magnetic properties of a metal salen complex as represented by the following general formula in order to magnetize the intended drug by...
US-9,505,731 Epoxide compound
A novel low viscosity epoxide having the following general Structure (I): Structure (I) wherein R1 and R2 can be, but is not limited to, hydrogen or a...
US-9,505,730 Mineralocorticoid receptor antagonists
The present invention is directed to compounds of the Formula I ##STR00001## as well as pharmaceutically acceptable salts thereof, that are potentially useful...
US-9,505,729 Isoxazole analogs as mediators of transcriptional induction of E-cadherin
In one aspect, the invention relates to N-((arylamino)alkyl)-5-arylisoxazole-3-carboxamide analogs, derivatives thereof, and related compounds, which are useful...
US-9,505,728 Triazolone compounds and uses thereof
The invention disclosed herein is directed to compounds of Formula (I) and pharmaceutically acceptable salts thereof, which are useful in the treatment of...
US-9,505,727 Rufinamide and derivatives and their use in modulating the gating process of human voltage-gated sodium channels
The present invention provides compounds of formula I which are capable of inhibition of the activation of hNav1.1 or hNav1.6 sodium channels in neurons....
US-9,505,726 Substituted biphenyl amides as P2X.sub.3 and P2X.sub.2/3 antagonists
Compounds of the formula I: ##STR00001## or a pharmaceutically acceptable salt thereof, wherein, R.sup.1 is optionally substituted phenyl or optionally...
US-9,505,725 Crystalline and mesomorphous forms of an AKT inhibiting pyrimidinyl-cyclopentane compound, compositions and...
Disclosed is (S)-2-(4-chlorophenyl)-1-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cy- clopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-(isopropylamino)propan-1-one ...
US-9,505,724 4-amino substituted condensed pyrimidine compounds as PDE4 inhibitors
The invention relates to novel substituted condensed pyrimidine compounds of general formula (I) ##STR00001## in which the chemical groupings, substituents...
US-9,505,723 Compound, dispersant and toner
The present invention provides a dispersant excellent in the solubility to a solvent, the adsorption power to a coloring material, and the coloring material...
US-9,505,722 Azepane derivatives and methods of treating hepatitis B infections
Provided herein are compounds useful for the treatment of HBV infection in a subject in need thereof, pharmaceutical compositions thereof, and methods of...
US-9,505,721 Aromatic imide compound and method for producing same
[Problem] to provide an aromatic imide compound wherein the sensitivity for visible light such as g-line, h-line etc. is increased and solubility is also...
US-9,505,720 Phenol derivatives and pharmaceutical or cosmetic use thereof
The present invention relates to novel compounds of general formula: ##STR00001## and to the cosmetic or pharmaceutical use thereof.
US-9,505,719 Synthesis and use of kinase inhibitors
An improved synthesis of a class of inhibitor of Focal Adhesion Kinase (FAK) is provided, wherein use of an expensive palladium-based catalyst is reduced and...
US-9,505,718 3-piperidone compounds and their use as neurokinin-1 (NK1) receptor antagonists
The invention relates to 3-piperidone compounds, and in particular, to (2S)-phenyl-3-piperidone and its synthesis method. Use of the thus-synthesized...
US-9,505,717 Acetic acid ester compound or salt thereof
An acetic acid ester compound represented by the following formula (I) or a salt thereof, ##STR00001## wherein R represents optionally substituted deuterated...
US-9,505,716 Pyrrolidine triple reuptake inhibitors
In various embodiments, the present invention provides cycloalkyl pyrrolidine compounds and methods for their use in the treatment and/or prevention of various...
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