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Patent # Description
US-9,512,109 Agonists that enhance binding of integrin-expressing cells to integrin receptors
A method of enhancing binding of cells to an integrin-binding ligand comprises treating integrin-expressing cells in vitro with an agonist of integrin, wherein...
US-9,512,108 9,9,10,10-Tetrafluoro-9,10-dihydrophenanthrene hepatitis C virus inhibitor and application thereof
The present invention belongs to the field of chemical pharmaceuticals, and specifically relates to compounds represented by formula I having a ...
US-9,512,107 Therapeutically active compositions and their methods of use
Provided are compounds useful for treating cancer and methods of treating cancer comprising administering to a subject in need thereof a compound described herein.
US-9,512,106 Smoothened modulators and methods of use thereof
Compounds of general Formulas (I), (IA), (IB) are described, along with compositions containing the same and methods of use thereof, inhibiting the hedgehog...
US-9,512,105 1-substituted 4-arylpiperazine as kappa opioid receptor antagonists
Provided are compounds represented by the formula: where R, Y.sub.3, R.sub.1, R.sub.2, R.sub.3, R.sub.4, R.sub.6, G, R.sub.7, E.sub.1, E.sub.2, A, B, W, X, Y...
US-9,512,104 Quinolone inhibitors of lipoprotein-associated phospholipase A2
The present invention relates to new quinolone inhibitors of lipoprotein-associated phospholipase A2 activity, pharmaceutical compositions thereof, and methods...
US-9,512,103 Synthesis of thiohydantoins
A novel synthesis of the anti-androgen, A52, which has been found to be useful in the treatment of prostate cancer, is provided. A52 as well as structurally...
US-9,512,102 4,6-difluorodibenzothiophene derivatives
4,6-difluorodibenzothiophene compounds of formula I ##STR00001## the preparation thereof, the use thereof as components in liquid-crystalline media and...
US-9,512,101 Beta- and gamma-amino-isoquinoline amide compounds and substituted benzamide compounds
Disclosed are beta and gamma-amino isoquinoline amide compounds and substituted benzamide compounds. In particular, the invention provides compounds that affect...
US-9,512,100 Method for producing glycolide
A method for producing glycolide (GL) by heating a glycolic acid oligomer (GAO) to depolymerize the GAO. The method for producing GL comprises: a step 1 of...
US-9,512,099 Compounds for inhibition of memapsin 1
Various embodiments of the present invention relate to, among other things, compounds that are inhibitors of Memapsin 1 and, as a result, are effective in the...
US-9,512,098 Process of producing purified gamma- and delta-tocotrienols from tocol-rich oils or distillates
The invention is generally directed to a process of producing purified gamma- and/or delta-tocotrienols from tocol-rich oils or distillates, such as rice bran...
US-9,512,097 Process for the preparation of 3-aroyl-5-aminobenzofuran derivatives
The present invention relates to a process for the preparation of 3-aroyl-5-aminobenzofuran derivatives useful as antiarrhythmic drugs which avoids the use of...
US-9,512,096 Synthesis of amine substituted 4,5,6,7-tetrahydrobenzothiazole compounds
The present invention is related to an improved process for the preparation of amino-substituted 4,5,6,7-tetrahydrobenzothiazole compounds of formula I, such as...
US-9,512,095 Polymorph forms of desazadesferrithiocin analogs
The present invention provides a solid form and compositions thereof, which are useful as metal chelators and which exhibit desirable characteristics for the same.
US-9,512,094 C17-heteroaryl derivatives of oleanolic acid and methods of use thereof
Disclosed herein are novel C17-heteroaryl derivatives of oleanolic acid, including those of the formula: ##STR00001## wherein the variables are defined...
US-9,512,093 Process for manufacturing 4-propargylated amino-benzoxazinones
The present invention relates to a process for manufacturing 4-propargylated amino-benzoxazinones of formula (I), ##STR00001## comprising the following steps:...
US-9,512,092 Retinoic acid receptor antagonists as chaperone-mediated autophagy modulators and uses thereof
Compounds, compositions and methods are provided for selectively activating chaperone-mediated autophagy (CMA), protecting cells from oxidative stress,...
US-9,512,091 Compositions and methods for the modulation of specific amidases for N-acylethanolamines for use in the therapy...
The present invention regards compositions and methods for the modulation of amidases capable of hydrolyzing N-acylethanolamines useable in the therapy of...
US-9,512,090 Tetrazolinone compound and use thereof
A tetrazolinone compound represented by formula (1): ##STR00001## Wherein R.sup.1, R.sup.2, R.sup.3, and R.sup.11 each represents a halogen atom, a C1-C6 alkyl...
US-9,512,089 Tetrazole-substituted arylamides as P2X.sub.3 and P2X.sub.2/3 antagonists
Compounds of the formula I: ##STR00001## or a pharmaceutically acceptable salt thereof, wherein, R.sup.1 is optionally substituted tetrazolyl, R.sup.2 is...
US-9,512,088 Method for producing N-sulfonyl-substituted oxindoles
Process for the selective N-sulfonylation of oxindoles, in particular process for the N-sulfonylation of 3-triazinyloxindoles, and also N-sulfonyl-substituted...
US-9,512,087 Hybrid molecules containing pharmacophores of fluconazole as antifungal agents and their preparation
Disclosed herein are novel antifungal compounds of Formula 1, containing fluconazole pharmacophore moieties coupled with other moieties including aryl enones...
US-9,512,086 Compound for promoting apoptosis of cancer cells and a pharmaceutical composition containing the same and uses...
The present invention provides a compound of Formula (I) and a salt thereof, ##STR00001## wherein, m is an integer of 2 to 7, and R is independently at...
US-9,512,085 Salts of a dihydroquinazoline derivative
The invention relates to besylate and tosylate salts of {8-fluoro-2-[4-(3-methoxyphenyl)piperazin-1-yl]-3-[2-methoxy-5-(trifluoro- ...
US-9,512,084 Amino pyrimidine derivatives
The present invention describes new amino pyrimidine derivatives and pharmaceutically acceptable salts thereof which appear to interact with Bruton's tyrosine...
US-9,512,083 Histone deacetylase 6 selective inhibitors for the treatment of bone disease
This invention relates to methods for treating bone disease associated with osteoclast activation using HDAC6 selective inhibitors, e.g., small molecule...
US-9,512,082 Inhibitors of glutaminyl cyclase
Compounds of formula (I), combinations and uses thereof for disease therapy, ##STR00001## or a pharmaceutically acceptable salt, solvate or polymorph...
US-9,512,081 Process for preparing 3,5-bis(fluoroalkyl)pyrazole derivatives from .alpha.,.alpha.-dihaloamines
The present invention relates to a novel process for preparing 3,5-bis(fluoroalkyl)pyrazole derivatives from .alpha.,.alpha.-dihaloamines.
US-9,512,080 Synthesis of acridinium compounds by N-alkylation of acridans
A method is provided for N-alkylation of acridine compounds by reduction of acridines to corresponding acridans to improve the reactivity of the acridine...
US-9,512,079 Deuterated CFTR potentiators
This invention relates to compounds of Formula I: ##STR00001## and pharmaceutically acceptable salts thereof. This invention also provides compositions...
US-9,512,078 Process for preparing 3-[(45)-8-bromo-1-methyl-6-(2-pyridinyl)-4H-imidazo[1,2-A][1,4]benzodiaze- ...
The invention concerns a new process for preparing 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4H-imidazo[1,2-a][1,4]benzodiaze- pine-4-yl]-propionic acid methyl...
US-9,512,077 Process for the preparation of methylphenidate hydrochloride and its intermediates thereof
The present invention relates to an industrially feasible and economically viable process for the preparation of methylphenidate hydrochloride of formula I and...
US-9,512,076 Indirubin derivatives and uses thereof in treating chronic myelogenous leukemia
Indirubin is the major active anti-tumor component of a traditional Chinese herbal medicine used for treatment of chronic myelogenous leukemia (CML). One aspect...
US-9,512,075 Compound; tautomer and geometric isomer thereof; salt of said compound, tautomer, or geometric isomer; method...
The present invention provides compounds belonging to 3-acyloxyindole compounds or 3-acyl-4-hydroxycoumarin compounds, a tautomer or geometric isomer thereof,...
US-9,512,074 Radiolabeled inhibitors of the amino acid transporters ASCT1 and ASCT2
The present invention relates to a compound of Formula (I) or (II) ##STR00001## or a salt thereof, wherein R is described herein. The compounds are novel...
US-9,512,073 Amino acid-, peptide-and polypeptide-lipids, isomers, compositions, and uses thereof
Described herein are compounds and compositions characterized, in certain embodiments, by conjugation of various groups, such as lipophilic groups, to an amino...
US-9,512,072 Biodegradable computed tomography contrast agents
Biodegradable computed tomography (CT) contrast agents comprising a polyiodinated aryl contrast agent that is crosslinked by an organic disulfide are described...
US-9,512,071 Mixed decyl mercaptans compositions and methods of making same
Compositions comprising branched C.sub.10 mercaptans selected from the group consisting of 5-methyl-1-mercapto-nonane, 3-propyl-1-mercapto-heptane,...
US-9,512,070 Method for producing compound containing BIS (perfluoroalkylsulfonyl) methyl group and salt thereof, and solid...
A method for producing compounds containing a bis(perfluoroalkylsulfonyl)methyl group or salts thereof, wherein the compounds have high acidity and...
US-9,512,069 Urea synthesis process and plant
Disclosed is a urea plant comprising an additional reactor. With reference to the regular components of a urea plant, including a recovery section and a high...
US-9,512,068 Augmenting moieties for anti-inflammatory compounds
Augmented or synergized anti-inflammatory constructs are disclosed including terpenes covalently conjugated with other anti-inflammatory molecules such as...
US-9,512,067 Method for producing xylylene diisocyanate and system for producing xylylene diisocyanate
A method for producing xylylene diisocyanate includes a thermal decomposition step of thermally decomposing xylylene dicarbamate; a first separation step of...
US-9,512,066 Enhancers of protein degradation
The present invention relates to compounds suitable for modulating huntingtin protein processing and useful for treating or preventing huntingtin-related...
US-9,512,065 Polymorphs of N-[(R)-1-[(S)-1-(4-aminomethyl-benzylcarbamoyl)-2-phenyl-ethylcarbamoyl]-- ...
The invention provides new polymorphs of N--[(R)-1-[(S)-1-(4-aminomethyl-benzylcarbamoyl)-2-phenyl-ethylcarbamoyl]- -2-(4-ethoxy-phenyl)-ethyl]-benzamide...
US-9,512,064 Tranilast compositions and cocrystals
Mew tranilast complexes and new tranilast cocrystais are disclosed. These include all tranilast nicotinamide complex, a 1:1 tranilast nicotinamide cocrystal, a...
US-9,512,063 Process for the preparation of advantame
A novelprocess for the preparation of N--[N-[3-(3-hydroxy-4-methoxyphenyl)-propyl]-L-.alpha.-aspartyl]-L-phenyl- alanine-1-methyl ester is described. It...
US-9,512,062 Method for producing N-isopropyl(meth)acrylamide
A novel process is described which allows N-isopropyl(meth)acrylamide to be obtained in high purity and yield in a simple manner, by reacting methacrylic...
US-9,512,061 Process for the preparation of racemic alpha-amino acids
Process for the preparation of racemic .alpha.-amino acids or of glycine, wherein the corresponding .alpha.-hydroxycarboxylic acid, selected from hydroxyacetic...
US-9,512,060 Solid state forms of tapentadol salts
Provided herein are novel solid state forms of tapentadol salts, process for their preparation, pharmaceutical compositions, and method of treating thereof. The...
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