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Patent # Description
US-9,605,003 Heterocyclic compounds and uses thereof
Substituted bicyclic heterocyclic compounds such as isoquinolinone compounds and pharmaceutical compositions that modulate kinase activity, including PI3 kinase...
US-9,605,002 5,5-heteroaromatic anti-infective compounds
The invention provides a series of 5,5-heteroaromatic compounds, syntheses thereof, compositions thereof, and methods of using such compounds and compositions....
US-9,605,001 Production of polyketides and other natural products
The present invention relates to production of polyketides and other natural products and to libraries of compounds and individual novel compounds. One...
US-9,605,000 Spiro azetidine isoxazole derivatives and their use as SSTR antagonists
Provided is a compound represented by the following formula (1) or a salt thereof, which has an SSTR5 antagonistic action: wherein each symbol has the same...
US-9,604,999 Compounds and uses thereof for the modulation of hemoglobin
Provide herein are compounds and pharmaceutical compositions suitable as modulators of hemoglobin, methods and intermediates for their preparation, and methods...
US-9,604,998 Inhibitors of the renal outer medullary potassium channel
The present invention provides compounds of Formula I ##STR00001## and the pharmaceutically acceptable salts thereof, which are inhibitors of the ROMK...
US-9,604,997 Peri-carbinols
The present invention is directed to compounds of formula (I): ##STR00001## pharmaceutical compositions, and methods of use for treating, reducing a symptom of...
US-9,604,996 Cyclic thienouracil-carboxamides and use thereof
The present application relates to novel 2,4-dioxo-1,2,3,4-tetrahydrothieno[2,3-d]pyrimidine-6-carboxamide derivatives ("thienouracil"-carboxamides), to...
US-9,604,995 Process for the preparation of olanzapine pamoate
An improved process for preparation of Olanzapine pamoate monohydrate from Olanzpaine is disclosed which comprises mixing at room temperature a solution of...
US-9,604,994 Thienopyrimidine inhibitors of atypical protein kinase C
The present application provides a compound of formula (I) ##STR00001## or a salt thereof, wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, A, G,...
US-9,604,993 Intermediates and methods for the synthesis of halichondrin B analogs
Methods of synthesizing intermediates useful for the synthesis of halichondrin B analogs are described.
US-9,604,992 Compounds of dibenzylidene sorbitol ester type, process of preparation, use, compositions comprising them and...
The invention relates to novel compounds of dibenzylidene sorbitol ester type corresponding to the following formulae (I) and (II): ##STR00001## in which: R,...
US-9,604,991 Preparation method of ticagrelor and intermediates thereof
Disclosed in the present invention is a method for preparing Ticagrelor (I), comprising the following steps: a cyclization reaction of ...
US-9,604,990 Crystalline forms of pemetrexed diacid and manufacturing processes therefor
Crystalline forms of pemetrexed diacid are provided (Forms 1 and 2) which are readily produced for either laboratory-scale or industrial scale. Processes for...
US-9,604,989 Imidazopyridazines as Akt kinase inhibitors
The present invention relates to a method for the treatment of a cancer that is sensitive to Pi3K/Akt pathway inhibition by administering a therapeutically...
US-9,604,988 Agent for treating or inhibiting recurrence of acute myeloid leukemia
This invention relates to an agent for treating or inhibiting recurrence of acute myeloid leukemia and an agent for inhibiting growth of leukemia stem cells...
US-9,604,987 Synthesis of autophagy inducing compound and the uses thereof
The present invention relates to a composition comprising compound of formula CB6 or CB8, ##STR00001## the pharmaceutically-acceptable carrier, solvent, the...
US-9,604,986 Polymorphs and process for preparation of (2S, ...
A process for preparation of compound of Formula (I) is disclosed. The application is also directed to polymorphic forms of the compound of formula (I). ...
US-9,604,985 Process for the preparation of chiral tert-butyl ...
A process for the preparation of N-protected 6-(piperidin-4-ylcarbamoyl)piperidin-3-yl sulfonates of Formula (III): which comprises contacting a lactone of...
US-9,604,984 5-chloro-2-difluoromethoxyphenyl pyrazolopyrimidine compounds, compositions and methods of use thereof
Compounds of Formula (00A) and methods of use as Janus kinase inhibitors are described herein.
US-9,604,983 Herbicidal 3-(2-benzyloxyphenyl)-2,4-dihydroxy-1,8-naphthyridine derivatives
The present invention relates to herbicidal benzyloxy-substituted phenyl-diones and phenyl-dioxo-thiazinones of formula (I), as well as to herbicidal...
US-9,604,982 P2X7 modulators
The present invention is directed to a compound of Formula (I) or (Ia) ##STR00001## The invention also relates to pharmaceutical compositions comprising...
US-9,604,981 IP receptor agonist heterocyclic compounds
The present invention provides heterocyclic derivatives of formula (Ia) which activate the IP receptor. Activating the IP receptor signaling pathway is useful...
US-9,604,980 Substituted pyrimidinyl and pyridinyl-pyrrolopyridinones, process for their preparation and their use as kinase...
The present invention relates to substituted pyrimidinyl- and pyridinylpyrrolopyridinone compounds which modulate the activity of protein kinases and are...
US-9,604,979 Pyrroloquinoline quinone alcohol adduct
The present invention relates to a compound represented by the formula (A) or (B), or a salt thereof capable of improving a red color of pyrroloquinoline...
US-9,604,978 Compounds for inflammation and immune-related uses
The invention relates to certain compounds or pharmaceutically acceptable salts, solvates, clathrates, or prodrugs thereof, that are useful as immunosuppressive...
US-9,604,977 Bicyclic thiophenylamide compounds
Compounds having the formula (I) ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, R.sup.7, A, E and n are as described herein,...
US-9,604,976 Antibacterial compounds
The present invention provides a compound of the following formula, salts, racemates, diastereomers, enantiomers, esters, carbamates, phosphates, sulfates,...
US-9,604,975 Indolyl-pyridone derivatives having checkpoint kinase 1 inhibitory activity
Compounds of formula (I) have checkpoint kinase 1 (CHK1) inhibitory activity: ##STR00001## wherein R.sub.1, R.sub.2, R.sub.5 and R.sub.6 are independently...
US-9,604,974 Compounds as modulator of JAK-STAT pathway, methods and applications thereof
The present disclosure relates to compound of structural Formula I and a method for preparing said compounds. The disclosure further relates to a method of...
US-9,604,973 Anti-cancer polyketide compounds
Provided herein, inter alia, are anticancer polyketides. The uses of the polyketides described herein include treatment of cancer, for example, through...
US-9,604,972 Nitrogen-containing heteroaromatic ring compound
A nitrogen-containing heteroaromatic compound is represented by the following formula (A). ##STR00001## wherein Y is an oxygen atom or a sulfur atom, M is a...
US-9,604,971 Co-crystal of the PAR-1 receptor antagonists vorapaxar and aspirin
This invention relates to a co-crystal of vorapaxar and aspirin. The inventive co-crystal antagonizes the PAR-1 receptor. This invention also provides for...
US-9,604,970 1,3-dihydroimidazole-2-thione derivatives for use in the treatment of pulmonary arterial hypertension and lung...
The present invention relates to compounds of formula I: ##STR00001## for use in treating pulmonary arterial hypertension and associated conditions, where...
US-9,604,969 Pyrimidin-4-yl)oxy)-1h-indole-1-carboxamide derivatives and use thereof
This invention relates to certain metabolites of N-(1-methyl-5-(trifluoromethyl)-1H-pyrazol-3-yl)-5-((6-((methyl-amino)met- ...
US-9,604,968 Pure crystalline Form II of L-malic acid salt of sunitinib and processes for its preparation
The present invention relates to pure crystalline Form II of an L-malic acid salt of sunitinib and a process for its preparation. The invention further provides...
US-9,604,967 Azetidinyloxyphenylpyrrolidine compounds
The invention provides certain azetidinyloxyphenylpyrrolidine compounds, particularly compounds of formula I wherein R is hydrogen or methyl, and pharmaceutical...
US-9,604,966 Crizotinib preparation method
The present invention relates to the technical field of medicine and organic synthesis, particularly to a method for preparing crizotinib. The method comprises...
US-9,604,965 Substituted pyridazines as skeletal muscle modulators
Provided are compounds of Formula I: ##STR00001## or a pharmaceutically acceptable salt thereof, wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6,...
US-9,604,964 Dihydropyrazole GPR40 modulators
The present invention provides compounds of Formula (I): (Formula (I), or a stereoisomer, or a pharmaceutically acceptable salt thereof, wherein all of the...
US-9,604,963 Amino-quinolines as kinase inhibitors
Disclosed are compounds having the formula: ##STR00001## wherein R.sup.1, R.sup.2, R.sup.3 and Z are as defined herein, and methods of making and using the...
US-9,604,962 Fungicidal azocyclic amides
Disclosed are compounds of Formulae 1, 1A, 1B and 1C including all geometric and stereoisomers, N-oxides, and salts thereof, ##STR00001## wherein R.sup.1,...
US-9,604,961 Histone demethylase inhibitors
Provided herein are substituted pyrazolylpyridine, pyrazolylpyridazine, and pyrazolylpyrimidine derivative compounds and pharmaceutical compositions comprising...
US-9,604,960 Aryl, heteroaryl, and heterocycle substituted tetrahydroisoquinolines and use thereof
Novel aryl, heteroaryl, and non-aromatic heterocyle substituted tetrahydroisoquinolines are described in the present invention. These compounds are used in the...
US-9,604,959 Thiol compound and composition for optical materials using the same
According to the present invention, it is possible to provide a thiol compound represented by formula (1): ##STR00001## wherein R.sub.1 is ...
US-9,604,958 HIF inhibitors and use thereof
The present invention is directed to HIF inhibitors and methods of preventing cell proliferation, reducing inflammation, and treating an angiogenic disease or...
US-9,604,957 Selective matrix metalloproteinase inhibitors
The invention provides compounds, compositions, and methods for the treatment of diseases, disorders, or conditions that are modulated by matrix...
US-9,604,956 Process for the production of trioxane
The present invention relates to a process for producing cyclic acetal comprising i) preparing a liquid reaction mixture comprising a) formaldehyde source, b)...
US-9,604,955 Chemical enhancement by nanomaterials under X-ray irradiation
A method for dynamic enhancement of chemical reactions by nanomaterials under hard X-ray irradiation. The nanomaterials were gold and platinum nanoparticles,...
US-9,604,954 2,3-Fluorinated glycosides as neuraminidase inhibitors and their use as anti-virals
Compounds having a structure of Formula I and compositions comprising these compounds are provided. Uses of such compounds and compositions are provided for...
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